SCHEMBL24958720

SCHEMBL24958720

CSc1ccc(-n2cnc(C3CC3)n2)nc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
ACACB O00763 1/20 0.33
GRM5 P41594 2/20 0.30
GRM1 Q13255 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24958923 0.78 GRM5 (0.32) GRM5GRM1
SCHEMBL24958718 0.77 EGLN1 (0.35) ACACBGRM5GRM1
SCHEMBL24960023 0.72 MAPT (0.48) LMNA
SCHEMBL24908617 0.69 HDAC4 (0.32) OPRM1OPRL1
SCHEMBL19706489 0.68 OPRM1 (0.49) OPRM1OPRL1
SCHEMBL24960022 0.66 GPR119 (0.33) LMNA
SCHEMBL22144631 0.66 HRH3 (0.45) ACACBLMNA
SCHEMBL26674231 0.65 DHFR (0.45) OPRM1OPRL1ACACB
SCHEMBL28121336 0.65
SCHEMBL25326218 0.63 GRM5 (0.33) GRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230021705-A1 GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230021705-A1 GLP-1R MODULATING COMPOUNDS GLP1R, GIPR, GPR119 OPRM1 1503/4885OPRL1 393/4885ACACB 674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.