SCHEMBL249613

SCHEMBL249613

OCCc1ccc(N2CCOCC2)c(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.49
ALDH1A1 P00352 4/20 0.46
LMNA P02545 2/20 0.46
KDM4E B2RXH2 1/20 0.46
PDE3B Q13370 2/20 0.45
PDE3A Q14432 2/20 0.45
CYP2C9 P11712 1/20 0.44
AKR1C3 P42330 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
SRPK1 Q96SB4 1/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
GAA P10253 2/20 0.42
S1PR1 P21453 1/20 0.40
SLC6A9 P48067 1/20 0.40
PIK3CA P42336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12142079 0.83 NOTUM (0.51) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL250868 0.83 ALDH1A1 (0.51) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL250808 0.81 NOTUM (0.49) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL20716309 0.76 NPC1 (0.52) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL24680705 0.75 NOTUM (0.54) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL249879 0.75 NOTUM (0.58) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL1929073 0.75 MAPT (0.61) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL31210319 0.75 MAPT (0.61) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL29623590 0.75 NOTUM (0.54) NOTUMALDH1A1LMNAKDM4EPDE3B
SCHEMBL7911412 0.75 NOTUM (0.54) NOTUMALDH1A1LMNAKDM4EPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP disclosed
WO-2010097410-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS RESPIRATORIUS AB (SE) 2010-09-02 WO disclosed