SCHEMBL249879

SCHEMBL249879

[CH2]c1ccc(N2CCOCC2)c(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.58
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 2/20 0.51
LMNA P02545 1/20 0.51
PDE3B Q13370 2/20 0.49
PDE3A Q14432 2/20 0.49
AKR1C3 P42330 1/20 0.46
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
TP53 P04637 1/20 0.45
THRB P10828 1/20 0.45
S1PR1 P21453 1/20 0.44
PIK3R1 P27986 3/20 0.42
PIK3CA P42336 3/20 0.42
PIK3CD O00329 1/20 0.42
PIK3C2B O00750 1/20 0.42
PIK3CB P42338 1/20 0.42
MTOR P42345 1/20 0.42
PIK3CG P48736 1/20 0.42
PRKDC P78527 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249224 0.83 NOTUM (0.50) NOTUMALDH1A1PDE3BPDE3AS1PR1
SCHEMBL17102319 0.81 NOTUM (0.54) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL1929073 0.81 MAPT (0.61) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL7911412 0.81 NOTUM (0.54) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL31210319 0.81 MAPT (0.61) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL24680705 0.81 NOTUM (0.54) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL29623590 0.81 NOTUM (0.54) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL12433016 0.79 NOTUM (0.53) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL12139639 0.78 ALDH1A1 (0.56) NOTUMALDH1A1KDM4ELMNAPDE3B
SCHEMBL10232907 0.77 NOTUM (0.51) NOTUMALDH1A1KDM4ELMNAPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP claimed