SCHEMBL24967825

SCHEMBL24967825

COc1ccc([C@@H]2CN(C(=O)OCC3c4ccccc4-c4ccccc43)CC2C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FABP5 Q01469 2/20 0.43
PPARG P37231 3/20 0.43
PPARA Q07869 2/20 0.43
FABP7 O15540 1/20 0.42
PDE4B Q07343 3/20 0.42
EDNRA P25101 2/20 0.42
EDNRB P24530 1/20 0.42
MDM2 Q00987 1/20 0.42
ALDH1A1 P00352 2/20 0.41
FFAR1 O14842 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ACHE P22303 1/20 0.40
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24967824 0.90 FABP5 (0.51) FABP5PPARGPPARAFABP7PDE4B
SCHEMBL24967716 0.89 FABP5 (0.44) FABP5PPARGPPARAFABP7PDE4B
SCHEMBL24967216 0.87 FABP5 (0.44) FABP5PPARGPPARAFABP7MDM2
SCHEMBL24967215 0.87 FABP5 (0.44) FABP5PPARGPPARAFABP7MDM2
SCHEMBL24967724 0.87 FABP5 (0.44) FABP5PPARGPPARAFABP7PDE4B
SCHEMBL24967722 0.82 PPARG (0.47) FABP5PPARGPPARAFABP7PDE4B
SCHEMBL24967723 0.80 FABP5 (0.44) FABP5PPARGPPARAFABP7PDE4B
SCHEMBL24967230 0.79 EDNRA (0.38) FABP5PPARGPPARAFABP7EDNRA
SCHEMBL23924125 0.77 ALDH1A1 (0.48) PDE4BEDNRAEDNRBALDH1A1MEN1
SCHEMBL20475203 0.77 ALDH1A1 (0.48) PDE4BEDNRAEDNRBALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192340-A9 SMALL MOLECULE ALLOSTERIC MODULATORS OF CLASS B GPCR, THE PTHR, AND METHOD TO IDENTIFY THEM UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2023-02-02 WO disclosed