SCHEMBL24967945

SCHEMBL24967945

CC1CN(c2ncc(C(F)(F)F)cn2)CCN1C(=O)Oc1cccc(-c2c[nH]c(=O)c(C(F)(F)F)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 6/20 0.43
CHRM1 P11229 6/20 0.43
CHRM3 P20309 4/20 0.42
TRPA1 O75762 1/20 0.41
CHRM4 P08173 6/20 0.41
FAAH O00519 5/20 0.41
TIPARP Q7Z3E1 1/20 0.39
SLC6A9 P48067 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24967944 1.00 CHRM2 (0.43) CHRM2CHRM1CHRM3TRPA1CHRM4
SCHEMBL24967938 0.86 TRPA1 (0.54) TRPA1TIPARP
SCHEMBL30164987 0.86 TRPA1 (0.54) TRPA1TIPARP
SCHEMBL29165932 0.80 SLC6A9 (0.47) TIPARPSLC6A9
SCHEMBL29165852 0.79 TIPARP (0.40) CHRM4TIPARPSLC6A9
SCHEMBL24968205 0.79 TRPA1 (0.42) TRPA1TIPARP
SCHEMBL24967934 0.79 TRPA1 (0.42) TRPA1TIPARP
SCHEMBL24968206 0.79 TRPA1 (0.42) TRPA1TIPARP
SCHEMBL24968226 0.78 CHRM4 (0.45) CHRM2CHRM1CHRM3CHRM4TIPARP
SCHEMBL24968434 0.78 CHRM4 (0.45) CHRM2CHRM1CHRM3CHRM4TIPARP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006013-A1 NOVEL PARP7 INHIBITOR AND USE THEREOF 上海齐鲁制药研究中心有限公司 2023-02-02 WO disclosed