SCHEMBL24969699

SCHEMBL24969699

C[C@@H]1CN(c2nc3ccccc3nc2Cl)CCN1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.56
HTR3B O95264 1/20 0.56
HTR3A P46098 1/20 0.56
MAPT P10636 3/20 0.45
MAPK13 O15264 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
MAPK14 Q16539 1/20 0.43
TSHR P16473 2/20 0.41
TDP1 Q9NUW8 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GFER P55789 2/20 0.40
CSNK1E P49674 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
LMNA P02545 1/20 0.40
ADRA2A P08913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31142966 1.00 HRH4 (0.56) HRH4HTR3BHTR3AMAPTMAPK13
SCHEMBL24969701 1.00 HRH4 (0.56) HRH4HTR3BHTR3AMAPTMAPK13
Hydrochloric Acid SCHEMBL29268333 0.99 HRH4 (0.55) HRH4HTR3BHTR3AMAPTMAPK13
Hydrochloric Acid SCHEMBL30223438 0.82 ADRA2A (0.41) MAPTMAPK13MAPK12MAPK11MAPK14
SCHEMBL4307835 0.79 HTR3A (0.66) HRH4HTR3BHTR3AMAPTTSHR
SCHEMBL31143046 0.79 HTR3A (0.66) HRH4HTR3BHTR3AMAPTTSHR
SCHEMBL27934102 0.78 ALDH1A1 (0.42) HRH4HTR3BHTR3AMAPTTDP1
SCHEMBL17014815 0.78 GPR6 (0.52)
Hydrochloric Acid SCHEMBL30222871 0.77 HTR3A (0.64) HRH4HTR3BHTR3AMAPTTSHR
SCHEMBL3669381 0.77 MEN1 (0.55) HRH4MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed