SCHEMBL24970920

SCHEMBL24970920

Cc1c(Cl)ccc2cc(Cl)c(N3CCN(COC(C)(C)C)CC3)nc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP1 P29466 1/20 0.34
RAB9A P51151 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
GPR6 P46095 1/20 0.32
GRM2 Q14416 3/20 0.32
CNR2 P34972 4/20 0.31
CNR1 P21554 3/20 0.31
TRPV1 Q8NER1 1/20 0.31
DRD2 P14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31143036 0.77 CNR1 (0.47) MAPTALDH1A1POLBMEN1KMT2A
SCHEMBL31142946 0.75 ADRB1 (0.43) MAPTKDM4ENPC1ALDH1A1POLB
SCHEMBL24970936 0.75 ADRB1 (0.43) MAPTKDM4ENPC1ALDH1A1POLB
Hydrochloric Acid SCHEMBL30223275 0.74 ADRB1 (0.42) MAPTKDM4ENPC1ALDH1A1POLB
SCHEMBL24511557 0.68 SLC6A2 (0.42) MAPTALDH1A1RAB9AKMT2ADRD2
SCHEMBL24969920 0.63 CNR1 (0.49) KDM4EALDH1A1POLBMEN1KMT2A
SCHEMBL31143026 0.63 CNR1 (0.49) KDM4EALDH1A1POLBMEN1KMT2A
SCHEMBL31143096 0.62 PPARA (0.36) MAPTKDM4ENPC1ALDH1A1RAB9A
SCHEMBL24971015 0.62 PPARA (0.36) MAPTKDM4ENPC1ALDH1A1RAB9A
SCHEMBL23365940 0.61 MAPT (0.46) MAPTKDM4EALDH1A1ALOX15TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed