SCHEMBL24970936

SCHEMBL24970936

Cc1c(Cl)ccc2cc(Cl)c(N3CCNCC3)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.43
PDE10A Q9Y233 1/20 0.42
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
HTR3E A5X5Y0 2/20 0.40
HTR3B O95264 2/20 0.40
HTR3A P46098 2/20 0.40
HTR3D Q70Z44 2/20 0.40
HTR3C Q8WXA8 2/20 0.40
HRH4 Q9H3N8 4/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31142946 1.00 ADRB1 (0.43) ADRB1PDE10ACHRNB2CHRNA4HTR3E
Hydrochloric Acid SCHEMBL30223275 0.99 ADRB1 (0.42) ADRB1PDE10ACHRNB2CHRNA4HTR3E
SCHEMBL31142879 0.82 PIK3CD (0.50) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL24969941 0.82 PIK3CD (0.50) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL30222974 0.81 PIK3CD (0.49) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL24970920 0.75 MAPT (0.34) HRH4ALDH1A1MAPTHSD17B10TDP1
SCHEMBL31143036 0.73 CNR1 (0.47) ALDH1A1MAPTPOLBMEN1KMT2A
SCHEMBL4823755 0.72 ADRB1 (0.56) ADRB1CHRNB2CHRNA4HTR3EHTR3B
SCHEMBL24970932 0.72 TDP1 (0.54) ADRB1CHRNB2CHRNA4HTR3EHTR3B
SCHEMBL24969947 0.70 CHRNB2 (0.58) ADRB1CHRNB2CHRNA4HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed