SCHEMBL24970930

SCHEMBL24970930

N#Cc1cc2ccccc2nc1N1CCNCC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.57
KDM4E B2RXH2 8/20 0.50
ALDH1A1 P00352 6/20 0.50
TSHR P16473 4/20 0.50
CYP1A2 P05177 3/20 0.50
CYP3A4 P08684 3/20 0.50
TP53 P04637 3/20 0.50
MAPK1 P28482 3/20 0.50
TDP1 Q9NUW8 3/20 0.50
HPGD P15428 2/20 0.50
LMNA P02545 2/20 0.50
HSD17B10 Q99714 2/20 0.50
HTR6 P50406 2/20 0.50
USP2 O75604 2/20 0.50
CYP2D6 P10635 1/20 0.50
HTR3E A5X5Y0 1/20 0.50
HTR3B O95264 1/20 0.50
ADRB1 P08588 1/20 0.50
HTR1A P08908 1/20 0.50
HTR2C P28335 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31142938 1.00 TAAR1 (0.57) TAAR1KDM4EALDH1A1TSHRCYP1A2
Hydrochloric Acid SCHEMBL29268332 0.99 TAAR1 (0.56) TAAR1KDM4EALDH1A1TSHRCYP1A2
SCHEMBL19051440 0.83 RXFP1 (0.65) KDM4EALDH1A1TSHRTP53MAPK1
SCHEMBL29654298 0.82 PDE10A (0.46) TAAR1KDM4EALDH1A1TSHRTP53
Hydrochloric Acid SCHEMBL29013581 0.80 KMT2A (0.50) TAAR1KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL6770354 0.79 ADRB1 (0.56) KDM4EALDH1A1TSHRCYP1A2CYP3A4
SCHEMBL24969918 0.78 HTR3A (0.54) KDM4EALDH1A1CYP1A2CYP3A4MAPK1
SCHEMBL24971049 0.78 HTR6 (0.54) KDM4EALDH1A1CYP1A2CYP3A4MAPK1
SCHEMBL7377147 0.78 CYP1A2 (0.59) TAAR1KDM4EALDH1A1TSHRCYP1A2
SCHEMBL6225002 0.78 HTR6 (0.54) KDM4EALDH1A1CYP1A2CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023002011-A1 GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-01-26 WO disclosed