SCHEMBL24975461

SCHEMBL24975461

Cc1nc(C(F)(F)F)ccc1OC[C@H]1C[C@@H](N)C1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.35
SYK P43405 1/20 0.35
TGFBR1 P36897 1/20 0.34
PDE4B Q07343 7/20 0.34
PTGS2 P35354 3/20 0.34
PTGS1 P23219 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
PDE11A Q9HCR9 1/20 0.32
PDE10A Q9Y233 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
RBP4 P02753 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24976603 0.84 TGFBR1 (0.34) SYKTGFBR1PTGS2PTGS1CHRNB2
SCHEMBL24976635 0.80 SYK (0.36) SYKPTGS2PTGS1
SCHEMBL24975374 0.79 TRPV1 (0.37) PDE4B
SCHEMBL30469190 0.74 TGFBR1 (0.38) AAK1SYKTGFBR1PDE4B
SCHEMBL25211504 0.74 TGFBR1 (0.38) AAK1SYKTGFBR1PDE4B
SCHEMBL21492158 0.73 CHRNB2 (0.55) CHRNB2CHRNA4
SCHEMBL21492160 0.73 CHRNB2 (0.55) CHRNB2CHRNA4
SCHEMBL12958179 0.73 MCHR1 (0.40) AAK1TGFBR1PDE4B
Hydrochloric Acid SCHEMBL21491545 0.72 CHRNB2 (0.57) CHRNB2CHRNA4
SCHEMBL20869211 0.69 PDE4B (0.48) TGFBR1PDE4BPTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023005894-A1 INHIBITOR COMPOUND FOR WNT PATHWAY 杭州阿诺生物医药科技有限公司 2023-02-02 WO disclosed