SCHEMBL249819

SCHEMBL249819

O=Cc1cn(C(=O)O)c2cccc(I)c12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
IMPDH2 P12268 1/20 0.33
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
POLB P06746 1/20 0.31
APEX1 P27695 1/20 0.31
CTDSP1 Q9GZU7 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
ERN1 O75460 3/20 0.31
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
HSP90AA1 P07900 1/20 0.30
IDO1 P14902 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28492551 0.86 KMT2A (0.39) ALDH1A1IMPDH2CNR1CNR2POLB
SCHEMBL28495147 0.85 PTGS2 (0.43) ALDH1A1L3MBTL1POLBAPEX1CTDSP1
SCHEMBL15901985 0.81 ALDH1A1 (0.36) ALDH1A1IMPDH2POLBTDP1KDM4E
SCHEMBL1229812 0.81 ERN1 (0.42) ALDH1A1ERN1MEN1KMT2A
SCHEMBL15902473 0.81 ALDH1A1 (0.39) ALDH1A1IMPDH2L3MBTL1POLBAPEX1
SCHEMBL20503064 0.81 CYP2A6 (0.41) ALDH1A1IMPDH2CNR1CNR2L3MBTL1
SCHEMBL28490523 0.81 HPGD (0.38) ALDH1A1L3MBTL1POLBERN1KDM4E
SCHEMBL28489226 0.80 HTR2C (0.39) ALDH1A1L3MBTL1MEN1NPC1RAB9A
SCHEMBL249361 0.80 ERN1 (0.33) ALDH1A1IMPDH2L3MBTL1POLBAPEX1
SCHEMBL28495086 0.79 PTGS2 (0.46) POLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001308-A9 METHOD FOR SYNTHESIZING ERGOLINE ALKALOIDS FROM INDOLIC BICYCLIC COMPOUNDS BY DOUBLE CYCLIZATION, RESULTING MATERIALS, AND INTERMEDIATE MATERIALS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-03-22 WO disclosed
WO-2012001308-A1 METHOD FOR SYNTHESIZING ERGOLINE ALKALOIDS FROM INDOLIC BICYCLIC COMPOUNDS BY DOUBLE CYCLIZATION, RESULTING MATERIALS, AND INTERMEDIATE MATERIALS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-01-05 WO disclosed