SCHEMBL2500295

SCHEMBL2500295

CNNC(=O)CC(=O)NNC

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
KDM5C P41229 1/20 0.57
EGLN1 Q9GZT9 1/20 0.57
PHF8 Q9UPP1 1/20 0.57
KDM2A Q9Y2K7 1/20 0.57
MCL1 Q07820 1/20 0.33
LMNA P02545 1/20 0.33
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12213974 0.82 KDM4E (0.43) KDM4EKDM5CEGLN1PHF8KDM2A
SCHEMBL2242250 0.80
SCHEMBL6773592 0.80
SCHEMBL12725535 0.80
SCHEMBL18576296 0.80
Hydrochloric Acid SCHEMBL2227956 0.78
Hydrochloric Acid SCHEMBL15414360 0.78
SCHEMBL16807522 0.78
SCHEMBL1750673 0.78
SCHEMBL6124941 0.78 KDM4E (0.64) KDM4EKDM5CEGLN1PHF8KDM2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021044884-A1 CURABLE RESIN COMPOSITION, SEALING AGENT FOR LIQUID CRYSTAL DISPLAY ELEMENT, VERTICALLY CONDUCTIVE MATERIAL, AND LIQUID CRYSTAL DISPLAY ELEMENT 積水化学工業株式会社 2021-03-11 WO disclosed
US-9156783-B2 Compounds for treating proliferative disorders SYNTA PHARMACEUTICALS CORP. (US) 2015-10-13 US disclosed
US-20150025042-A1 Compounds For Treating Proliferative Disorders SYNTA PHARMACEUTICALS CORP. (US) 2015-01-22 US disclosed
US-20130338162-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. (US) 2013-12-19 US disclosed
US-8609720-B2 Compounds for treating proliferative disorders SYNTA PHARMACEUTICALS CORP. (US) 2013-12-17 US disclosed
US-8497272-B2 Compounds for treating proliferative disorders SYNTA PHARMACEUTICALS CORP. (US) 2013-07-30 US disclosed
US-8383133-B2 Conjugates of Plasmodium falciparum surface proteins as malaria vaccines THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2013-02-26 US disclosed
US-20110245262-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. 2011-10-06 US disclosed
US-20100183678-A1 CONJUGATES OF PLASMODIUM FALCIPARUM SURFACE PROTEINS AS MALARIA VACCINES The Govenment of the United States of America as represented by tge Secreatary of Health (US) 2010-07-22 US disclosed
US-20100081635-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. 2010-04-01 US disclosed
EP-2074097-A2 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS Synta Pharmaceuticals Corporation (US) 2009-07-01 EP disclosed
EP-2057117-A2 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS Synta Pharmaceuticals Corporation (US) 2009-05-13 EP disclosed
WO-2008024303-A2 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. (US) 2008-02-28 WO disclosed
WO-2008024302-A2 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. (US) 2008-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100081635-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS HSPB1, HSP90AB1, HSPA1B KDM4E 3072/4885KDM5C 2631/4885EGLN1 4300/4885
US-20110245262-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS HSP90AB1, HSF1, HSP90B1 KDM4E 4105/4885KDM5C 3649/4885EGLN1 4564/4885
US-20100183678-A1 CONJUGATES OF PLASMODIUM FALCIPARUM SURFACE PROTEINS AS MALARIA VACCINES CD4, RPS25, OSBP2 KDM4E 4237/4885KDM5C 3071/4885EGLN1 2356/4885
US-20150025042-A1 Compounds For Treating Proliferative Disorders HSP90AB1, HSPB1, HSP90AB2P KDM4E 3309/4885KDM5C 3183/4885EGLN1 4500/4885
US-20130338162-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS HSP90AB1, HSF1, HSP90B1 KDM4E 4105/4885KDM5C 3649/4885EGLN1 4564/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.