SCHEMBL25005668

SCHEMBL25005668

CCS(=O)(=O)Nc1ccccc1Nc1ccnc(Cl)n1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.44
AURKA O14965 7/20 0.44
AURKB Q96GD4 3/20 0.44
MAPK8 P45983 6/20 0.41
SYK P43405 1/20 0.40
EGFR P00533 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MRGPRX1 Q96LB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31147659 1.00 PSIP1 (0.44) PSIP1AURKAAURKBMAPK8SYK
SCHEMBL30942621 0.91 AURKA (0.41) AURKAAURKBMAPK8SYKPTGS1
SCHEMBL27237965 0.91 AURKA (0.41) AURKAAURKBMAPK8SYKPTGS1
SCHEMBL30942599 0.86 PTGS1 (0.49) AURKAAURKBSYKEGFRPTGS1
SCHEMBL1039841 0.86 PTGS1 (0.49) AURKAAURKBSYKEGFRPTGS1
SCHEMBL30942660 0.81 SLC40A1 (0.50) AURKAAURKB
SCHEMBL5393403 0.80 MAPK14 (0.50) AURKAAURKBMAPK8SYKEGFR
SCHEMBL31147661 0.80 LMNA (0.52) AURKAAURKBALDH1A1LMNAHTT
SCHEMBL27238045 0.80 LMNA (0.52) AURKAAURKBALDH1A1LMNAHTT
SCHEMBL31147654 0.77 ALK (0.46) PSIP1MAPK8EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4382514-A1 PYRIMIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME AS ACTIVE INGREDIENT Korea Research Institute of Chemical Technology (KR) 2024-06-12 EP disclosed
WO-2023014022-A1 PYRIMIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME AS ACTIVE INGREDIENT 한국화학연구원 2023-02-09 WO disclosed