SCHEMBL25007019

SCHEMBL25007019

CC1(c2ccc(I)cc2)CNC(=O)C1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.41
OPRM1 P35372 2/20 0.36
OPRL1 P41146 1/20 0.36
CYP19A1 P11511 1/20 0.34
HTR6 P50406 1/20 0.33
CNR1 P21554 4/20 0.33
TDP2 O95551 2/20 0.31
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE1C Q14123 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12898108 0.81 OPRM1 (0.51) SMN1; SMN2OPRM1OPRL1
SCHEMBL9409501 0.74 MAPT (0.45) SMN1; SMN2
SCHEMBL2283567 0.71 AR (0.41) SMN1; SMN2OPRM1OPRL1
SCHEMBL16971269 0.70 OPRM1 (0.38) SMN1; SMN2OPRM1OPRL1CYP19A1TDP2
SCHEMBL25245033 0.69 OPRM1 (0.40) OPRM1HTR6
SCHEMBL31316550 0.68 OPRD1 (0.44)
SCHEMBL11659909 0.68 SMN1; SMN2 (0.41) SMN1; SMN2OPRM1OPRL1PDE1APDE1B
SCHEMBL11840395 0.68 CYP19A1 (0.34) CYP19A1HTR6CNR1TDP2
SCHEMBL29036149 0.66 OPRM1 (0.38) OPRM1
SCHEMBL665550 0.65 KCNH2 (0.46) OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117751113-A Aromatic acetylene derivative and preparation method and application thereof 浙江海正药业股份有限公司 2024-03-22 CN disclosed
WO-2023011573-A1 AROMATIC ACETYLENE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江海正药业股份有限公司 2023-02-09 WO disclosed
WO-2023011573-A1 AROMATIC ACETYLENE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江海正药业股份有限公司 2023-02-09 WO disclosed