SCHEMBL250129

SCHEMBL250129

NCCc1ccc(Br)cc1.O=C(O)NCCc1ccc(Br)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.60
HTR2A P28223 1/20 0.60
PLAAT3 P53816 2/20 0.51
PLAAT5 Q96KN8 2/20 0.51
PLAAT2 Q9NWW9 2/20 0.51
PLAAT4 Q9UL19 2/20 0.51
CNR1 P21554 1/20 0.49
MGLL Q99685 1/20 0.46
POLB P06746 3/20 0.46
CTDSP1 Q9GZU7 2/20 0.46
GRK2 P25098 2/20 0.46
LIG1 P18858 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
GPR35 Q9HC97 1/20 0.46
FPR2 P25090 1/20 0.46
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250873 0.91 PLAAT3 (0.58) TAAR1PLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL23111915 0.86 MCHR1 (0.50) TAAR1CNR1ALDH1A1KMT2A
SCHEMBL26988416 0.86 PLAAT3 (0.54) TAAR1PLAAT3PLAAT5PLAAT2PLAAT4
Phenethylcarbamic Acid SCHEMBL12478843 0.84 SMN1; SMN2 (0.59) TAAR1HTR2APLAAT3PLAAT5PLAAT2
SCHEMBL14672313 0.81 HSP90AA1 (0.58) PLAAT3PLAAT5PLAAT2PLAAT4CNR1
SCHEMBL915701 0.80 ESRRG (0.55) PLAAT3PLAAT5PLAAT2PLAAT4RAB9A
SCHEMBL16443753 0.80 KMT2A (0.52) PLAAT3PLAAT5PLAAT2PLAAT4CNR1
SCHEMBL5840627 0.79 CNR1 (0.54) TAAR1HTR2APLAAT3PLAAT5PLAAT2
SCHEMBL25303812 0.78 CNR1 (0.66) TAAR1PLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL5261796 0.78 MTNR1A (0.51) TAAR1HTR2APLAAT3PLAAT5PLAAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401275-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS Respiratorius AB (SE) 2012-01-04 EP disclosed
WO-2010097410-A1 NOVEL BRONCHODILATING DIAZAHETEROARYLS RESPIRATORIUS AB (SE) 2010-09-02 WO disclosed