SCHEMBL25035751

SCHEMBL25035751

CC(C)n1cc(-c2ccc(F)cn2)c(=O)c(C(=O)O)n1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F12 P00748 1/20 0.35
KMT2A Q03164 1/20 0.33
NTRK1 P04629 11/20 0.33
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
DHODH Q02127 1/20 0.32
GRM5 P41594 1/20 0.32
ACHE P22303 1/20 0.32
EIF4E P06730 1/20 0.32
TGFBR1 P36897 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25035787 0.85 F12 (0.35) F12KMT2AADORA2AADORA1DHODH
SCHEMBL29155062 0.84 ADORA3 (0.46) KMT2AADORA2AADORA1
SCHEMBL21753512 0.82 KMT2A (0.39) KMT2AADORA2AADORA1ACHE
SCHEMBL23882469 0.77 MET (0.39) NTRK1DHODHEIF4E
SCHEMBL19207117 0.74 CSNK1D (0.44) DHODH
SCHEMBL25035782 0.72 CYP1A2 (0.39) KMT2AADORA2AADORA1
SCHEMBL29902500 0.72 ADORA2A (0.42) ADORA2AADORA1TGFBR1
SCHEMBL29155052 0.71 ADORA3 (0.43) ADORA2AADORA1
SCHEMBL25224762 0.70 GABRA5 (0.36) DHODHGRM5EIF4E
SCHEMBL30174181 0.70 GABRA5 (0.36) DHODHGRM5EIF4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117561260-A Heterocyclic compound, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2024-02-13 CN disclosed
WO-2023016296-A1 HETEROCYCLIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2023-02-16 WO disclosed