SCHEMBL25041348

SCHEMBL25041348

CC(C)(C)c1ccc(NC2CCC(N)CC2)c(C#N)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
CHEK1 O14757 4/20 0.35
ROCK2 O75116 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CCR6 P51684 2/20 0.34
GSK3B P49841 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1G2 P78368 1/20 0.32
KIF11 P52732 1/20 0.32
TNF P01375 1/20 0.32
CSNK2A2 P19784 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30279117 1.00 CDK2 (0.38) CDK2IRAK4CHEK1ROCK2MEN1
SCHEMBL25041354 0.81 ALDH1A1 (0.41) IRAK4ROCK2PDE3BPDE3ACSNK1D
SCHEMBL25041349 0.79 ROCK2 (0.37) CDK2ROCK2MAPKAPK2PDE3BPDE3A
SCHEMBL25041352 0.79 ROCK2 (0.49) IRAK4ROCK2PDE3BPDE3ACSNK1D
SCHEMBL30279151 0.73 CHEK1 (0.38) CDK2IRAK4CHEK1GSK3BMAPKAPK2
SCHEMBL25039462 0.73 CHEK1 (0.38) CDK2IRAK4CHEK1GSK3BMAPKAPK2
SCHEMBL25040031 0.71 EPHX1 (0.42) MEN1KMT2AKIF11
SCHEMBL25040038 0.71 EPHX1 (0.42) MEN1KMT2AKIF11
SCHEMBL25039545 0.71 EPHX1 (0.42) MEN1KMT2AKIF11
SCHEMBL19194279 0.71 KIF11 (0.39) MEN1KMT2ACSNK1DCSNK1G2KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118076581-A Iron death modulators, their preparation and use 维泰瑞隆有限公司 2024-05-24 CN disclosed
WO-2023016447-A1 FERROPTOSIS MODULATORS, PREPARATIONS, AND USES THEREOF Sironax Ltd. (KY) 2023-02-16 WO disclosed