SCHEMBL25045261

SCHEMBL25045261

CN1CCN2c3cccnc3NC(=O)C2C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.43
CYP1A2 P05177 3/20 0.43
CHRM2 P08172 3/20 0.43
CYP2D6 P10635 3/20 0.43
CHRM1 P11229 3/20 0.43
HTR2C P28335 3/20 0.43
HTR2B P41595 3/20 0.43
HTR1A P08908 2/20 0.43
ADRA2A P08913 2/20 0.43
CYP2C9 P11712 2/20 0.43
TSHR P16473 2/20 0.43
ADRA2B P18089 2/20 0.43
ADRA2C P18825 2/20 0.43
DRD1 P21728 2/20 0.43
CYP2C19 P33261 2/20 0.43
HTR7 P34969 2/20 0.43
ADRA1A P35348 2/20 0.43
HRH1 P35367 2/20 0.43
DRD3 P35462 2/20 0.43
HTR3A P46098 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27242701 0.81 OPRM1 (0.39) ALDH1A1OPRM1KDM4ESMN1; SMN2GSK3B
SCHEMBL25045262 0.79 CYP1A2 (0.52) HTR2ACYP1A2CHRM2CYP2D6CHRM1
SCHEMBL11453737 0.78 KDM4E (0.62) HTR2ACYP1A2CHRM2CYP2D6CHRM1
SCHEMBL11487740 0.77 HTR2C (0.51) HTR2ACYP1A2CYP2D6HTR2CHTR2B
SCHEMBL25045512 0.77 DTYMK (0.46) DDB1CRBN
SCHEMBL25043787 0.74 DRD2 (0.43) HTR2ACYP1A2CHRM2CYP2D6CHRM1
SCHEMBL25045260 0.74 KDM4E (0.41) HTR2ACYP1A2CHRM2CYP2D6CHRM1
SCHEMBL25045347 0.74 KDM4E (0.41) HTR2ACYP1A2CHRM2CYP2D6CHRM1
SCHEMBL31067329 0.73 GRIN2B (0.45) CYP2D6CYP2C9CYP2C19MEN1CYP3A4
SCHEMBL10280080 0.71 HTR2A (0.37) HTR2ACYP1A2CHRM2CYP2D6CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023016521-A1 SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 上海赛默罗生物科技有限公司 2023-02-16 WO disclosed