SCHEMBL25048619

SCHEMBL25048619

CC(C)(C)OC(=O)N(CCCN=O)Cc1ccc2ccccc2c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MC3R P41968 11/20 0.47
MC4R P32245 9/20 0.47
MC5R P33032 13/20 0.43
MC1R Q01726 2/20 0.40
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
NCOR2 Q9Y618 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
BCHE P06276 2/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30941017 0.87 MC3R (0.50) MC3RMC4RMC5RMC1RHDAC3
SCHEMBL3312799 0.87 MC3R (0.50) MC3RMC4RMC5RMC1RHDAC3
SCHEMBL13783897 0.85 CYP1A2 (0.54) MC3RMC4RMC5RMC1RHDAC3
SCHEMBL13783902 0.82 HDAC1 (0.58) MC3RMC4RHDAC3HDAC1HDAC2
SCHEMBL25047687 0.81 MC4R (0.44) MC3RMC4RMC5RMC1RHDAC3
SCHEMBL13783994 0.81 HDAC1 (0.65) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL26654244 0.80 MC4R (0.49) MC3RMC4RMC5RMC1RHDAC3
SCHEMBL26654243 0.80 MC4R (0.49) MC3RMC4RMC5RMC1RHDAC3
SCHEMBL31617921 0.78 SIGMAR1 (0.41) MC3RMC4RMC5RHDAC1SIGMAR1
SCHEMBL25046547 0.78 SIGMAR1 (0.41) MC3RMC4RMC5RHDAC1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023017152-A1 SPECIFIC SMALL MOLECULE INHIBITORS THAT BLOCK KMT9 METHYLTRANSFERASE ACTIVITY AND FUNCTION ALBERT-LUDWIGS-UNIVERSITÄT FREIBURG (DE) 2023-02-16 WO disclosed