SCHEMBL25066

SCHEMBL25066

CCCCCCc1[c]ccc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PTGS2 P35354 3/20 0.35
ESR1 P03372 2/20 0.35
ADRA2A P08913 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
TACR2 P21452 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
TP53 P04637 2/20 0.35
CYP3A4 P08684 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
SHBG P04278 1/20 0.35
HSPD1 P10809 1/20 0.35
ADRB3 P13945 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9330220 1.00 KCNH2 (0.38) KCNH2MEN1KMT2APTGS2ESR1
SCHEMBL5328557 0.98 MEN1 (0.37) KCNH2MEN1KMT2APTGS2TP53
SCHEMBL3595125 0.93 KMT2A (0.41) MEN1KMT2ASLC6A3TYR
SCHEMBL206972 0.85 MEN1 (0.33) MEN1KMT2A
SCHEMBL1940072 0.81 PTGS2 (0.37) KCNH2MEN1KMT2APTGS2ESR1
SCHEMBL1778766 0.80 PTGS2 (0.36) KCNH2MEN1KMT2APTGS2ESR1
SCHEMBL1778966 0.80 PTGS2 (0.44) PTGS2ESR1ADRA2AADORA3TACR2
SCHEMBL827972 0.80 PTGS2 (0.44) PTGS2ESR1ADRA2AADORA3TACR2
SCHEMBL283991 0.80 PTGS2 (0.44) PTGS2ESR1ADRA2AADORA3TACR2
SCHEMBL8709834 0.80 PTGS2 (0.36) KCNH2MEN1KMT2APTGS2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3558976-A1 SUBSTITUTED AZOLYLPYRROLONES AND AZOLYLHYDANTOINES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES Bayer CropScience Aktiengesellschaft (DE) 2019-10-30 EP disclosed
EP-2588480-A2 3,4-DIHYDROPYRROLO[1,2-A]PYRAZINE-2,8(1H)-DICARBOXAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF& xA; SANOFI (FR) 2013-05-08 EP disclosed
WO-2011161537-A2 3,4-DIHYDROPYRROLO[1,2-A]PYRAZINE-2,8(1H)-DICARBOXAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2011-12-29 WO disclosed
WO-1993023398-A1 SUBSTITUTED PYRIDO[1,2-A]PYRIMIDINONE DERIVATIVES AS FUNGICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-11-25 WO disclosed
EP-0027759-B1 SPIRO-DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM ETABLISSEMENTS NATIVELLE S.A. (FR) 1983-10-12 EP disclosed