SCHEMBL25075360

SCHEMBL25075360

CCOC(=O)c1ccc(Cl)[nH]c1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
MAPT P10636 2/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
LMNA P02545 2/20 0.57
GAA P10253 3/20 0.53
NPC1 O15118 1/20 0.53
POLB P06746 1/20 0.53
KDM4E B2RXH2 3/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.50
TSHR P16473 1/20 0.50
MDM2 Q00987 1/20 0.49
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8121938 0.83 ALDH1A1 (0.60) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL31032981 0.81 KDM4E (0.66) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL10004025 0.80 ALDH1A1 (0.57) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL18061496 0.78 ALDH1A1 (0.54) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL10748352 0.78 ALDH1A1 (0.58) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL4675224 0.77 ALOX15 (0.53) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL4899931 0.77 ALDH1A1 (0.50) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL18395324 0.77 TSHR (0.50) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL6375741 0.76 L3MBTL1 (0.53) ALDH1A1MAPTL3MBTL1LMNAGAA
SCHEMBL11372443 0.75 ALDH1A1 (0.51) ALDH1A1MAPTL3MBTL1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117377665-A PARP7 inhibitor and application thereof 北京华森英诺生物科技有限公司 2024-01-09 CN disclosed
WO-2023020479-A1 PARP7 INHIBITOR AND APPLICATION THEREOF 重庆华森制药股份有限公司 2023-02-23 WO disclosed