SCHEMBL25089907

SCHEMBL25089907

Cn1c(=O)c2[nH]c(-c3nc4ccccc4s3)nc2n(C)c1=O

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.61
KDM4E B2RXH2 2/20 0.61
ADORA2A P29274 2/20 0.61
CYP1A2 P05177 1/20 0.61
ADORA3 P0DMS8 1/20 0.61
ADORA1 P30542 1/20 0.61
BLM P54132 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
HSD17B10 Q99714 1/20 0.61
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
TDP1 Q9NUW8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
8-Phenyl Theophylline SCHEMBL516432 0.76 ADORA2A (1.00) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL25090497 0.75 KDM4E (0.61) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL25090488 0.74 KDM4E (0.67) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL28501882 0.74 ADORA1 (0.64) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL8596143 0.74 KDM4E (0.76) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL6868854 0.72 ADORA2B (0.76) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL25090354 0.72 KDM4E (0.72) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL2119734 0.72 KDM4E (0.72) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL10614178 0.72 KDM4E (1.00) ADORA2BKDM4EADORA2ACYP1A2ADORA3
SCHEMBL25090424 0.72 ADORA2B (0.63) ADORA2BKDM4EADORA2ACYP1A2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023023867-A1 COMPOUNDS FOR REDUCING CHOLESTEROL AND TREATING LIVER AND KIDNEY DISEASE MCMASTER UNIVERSITY (CA) 2023-03-02 WO disclosed