SCHEMBL28501882

SCHEMBL28501882

Cn1c(=O)c2[nH]c(-c3cccs3)nc2n(C)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.64
KDM4E B2RXH2 2/20 0.63
CYP1A2 P05177 1/20 0.63
ADORA3 P0DMS8 1/20 0.63
ADORA2A P29274 1/20 0.63
ADORA2B P29275 1/20 0.63
BLM P54132 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
HSD17B10 Q99714 1/20 0.63
ALDH1A1 P00352 1/20 0.57
HPGD P15428 1/20 0.57
TDP1 Q9NUW8 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9253597 0.87 ADORA1 (0.56) ADORA1KDM4ECYP1A2ADORA3ADORA2A
SCHEMBL25090614 0.77 ADORA2B (0.54) ADORA1KDM4ECYP1A2ADORA3ADORA2A
8-Phenyl Theophylline SCHEMBL516432 0.77 ADORA2A (1.00) ADORA1KDM4ECYP1A2ADORA3ADORA2A
SCHEMBL6868854 0.76 ADORA2B (0.76) ADORA1KDM4ECYP1A2ADORA3ADORA2A
SCHEMBL25090639 0.76 ADORA2B (0.67) ADORA1KDM4ECYP1A2ADORA3ADORA2A
SCHEMBL8596143 0.75 KDM4E (0.76) ADORA1KDM4ECYP1A2ADORA3ADORA2A
SCHEMBL25089897 0.74 ADORA2B (0.55) ADORA1KDM4ECYP1A2ADORA3ADORA2A
SCHEMBL25089907 0.74 ADORA2B (0.61) ADORA1KDM4ECYP1A2ADORA3ADORA2A
SCHEMBL9257595 0.74 ADORA2B (0.60) ADORA1KDM4ECYP1A2ADORA2AADORA2B
SCHEMBL10673069 0.74 KDM4E (0.64) ADORA1KDM4ECYP1A2ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111840298-A Application of small molecule inhibitor in preparing medicine for inhibiting interaction of ornithine decarboxylase and ornithine decarboxylase antitase 1 湖北工业大学 2020-10-30 CN claimed
CN-111840298-A Application of small molecule inhibitor in preparing medicine for inhibiting interaction of ornithine decarboxylase and ornithine decarboxylase antitase 1 湖北工业大学 2020-10-30 CN disclosed