SCHEMBL2510144

SCHEMBL2510144

N#Cc1ccc(-c2nc(N)ncc2NCCc2ccccc2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.44
ADORA2A P29274 1/20 0.44
CYP11B1 P15538 7/20 0.43
CYP11B2 P19099 7/20 0.43
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
RPS27 P42677 1/20 0.39
MAPK1 P28482 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ASPH Q12797 1/20 0.37
RIOX2 Q8IUF8 1/20 0.37
KDM8 Q8N371 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2500326 0.90 PRKACA (0.47) ADORA1ADORA2ACYP11B1CYP11B2CDK8
SCHEMBL2505744 0.81 ADORA1 (0.42) ADORA1ADORA2ACYP11B1CYP11B2
SCHEMBL1317568 0.77 HRH4 (0.52) ADORA2ACYP11B1CYP11B2RPS27SMN1; SMN2
SCHEMBL2521058 0.77 EGLN2 (0.39) CYP11B1CYP11B2
SCHEMBL2506224 0.76 PIK3CD (0.46) ADORA1ADORA2ACYP11B1CYP11B2
SCHEMBL2507060 0.76 CYP11B2 (0.44) ADORA1ADORA2ACYP11B1CYP11B2
SCHEMBL1998196 0.69 KDM4E (0.49) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL1317062 0.68 SMN1; SMN2 (0.55) CYP11B1CYP11B2CDK8MAPK1KDM4E
SCHEMBL22784143 0.68 CCNC (0.51) CCNCCDK8KDM4EALDH1A1MAPT
SCHEMBL29133731 0.66 EGFR (0.63) CCNCCDK8MAPK1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2362775-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2011-09-07 EP disclosed
WO-2010059658-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-05-27 WO disclosed