SCHEMBL25106975

SCHEMBL25106975

O=c1c(Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c(Nc2ccc3c(c2)CCC3)c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.48
RAPGEF4 Q8WZA2 2/20 0.48
NPC1 O15118 6/20 0.40
RAB9A P51151 6/20 0.40
TRPV1 Q8NER1 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
CASP3 P42574 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25106887 0.84 RAPGEF4 (0.41) KIF11RAPGEF4NPC1RAB9ATRPV1
SCHEMBL23933954 0.80 RAPGEF4 (0.58) RAPGEF4AKR1C3AKR1C2
SCHEMBL17423676 0.74 RAPGEF4 (0.49) RAPGEF4TRPV1AKR1C3AKR1C2
SCHEMBL24477512 0.71 TRPV1 (0.46) KIF11TRPV1MEN1KMT2A
SCHEMBL24477417 0.71 TRPV1 (0.46) KIF11TRPV1MEN1KMT2A
SCHEMBL379238 0.71 RAPGEF4 (0.63) RAPGEF4NPC1RAB9ASMN1; SMN2TP53
SCHEMBL17427531 0.71 RAPGEF4 (0.51) RAPGEF4AKR1C3AKR1C2
SCHEMBL15256134 0.71 RAPGEF4 (0.51) RAPGEF4AKR1C3AKR1C2
SCHEMBL23933952 0.70 RAPGEF4 (0.45) RAPGEF4
SCHEMBL15256120 0.69 RAPGEF4 (0.50) RAPGEF4AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023023882-A1 NITROGEN HETEROCYCLIC CARBENE-SQUARIC AMIDE BIFUNCTIONAL CATALYST AND PREPARATION METHOD THEREFOR 深圳湾实验室坪山生物医药研发转化中心 2023-03-02 WO disclosed