SCHEMBL25112474

SCHEMBL25112474

Cc1nc(OCC(F)(F)F)c2ccc(=O)n(C)c2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.35
SCN9A Q15858 2/20 0.34
PDE2A O00408 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
CNR2 P34972 1/20 0.34
RXRA P19793 1/20 0.34
MAPT P10636 2/20 0.32
ENPP1 P22413 1/20 0.32
RORC P51449 1/20 0.31
PTGS2 P35354 2/20 0.31
ADORA2A P29274 1/20 0.31
PTGS1 P23219 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCND2 P30279 1/20 0.31
CCND3 P30281 1/20 0.31
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23326799 0.78 ADORA1 (0.47) ADORA1CDK4CCND1CCND2CCND3
SCHEMBL25112473 0.73 CNR2 (0.36) CNR2LMNA
SCHEMBL30122255 0.69 MAT2A (0.42) ADORA1LMNA
SCHEMBL29861478 0.68 ADORA1 (0.41) ADORA1ADORA2ACDK4CCND1CCND2
SCHEMBL28863519 0.68 ADORA1 (0.39) ADORA1MAPTENPP1CDK4CCND1
SCHEMBL10042029 0.66 FADS1 (0.49) MAPTPTGS2TSHR
SCHEMBL25462029 0.63 CDK4 (0.55) ADORA1CDK4CCND1CCND2CCND3
SCHEMBL29861616 0.63 CDK4 (0.55) ADORA1CDK4CCND1CCND2CCND3
SCHEMBL24671864 0.63 ADORA1 (0.43) ADORA1MAPTENPP1CDK4CCND1
SCHEMBL29918643 0.63 ADORA1 (0.43) ADORA1MAPTENPP1CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4148056-A1 SOS1 INHIBITOR CONTAINING PHOSPHORUS CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2023-03-15 EP disclosed