SCHEMBL25148658

SCHEMBL25148658

COc1nc(-c2ccccc2OCC2CCOCC2)ccc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 4/20 0.43
PDCD1 Q15116 3/20 0.43
BRD4 O60885 2/20 0.41
PTGER1 P34995 1/20 0.40
XDH P47989 1/20 0.39
RIPK1 Q13546 1/20 0.39
DHFR P00374 1/20 0.39
DCPS Q96C86 1/20 0.39
BRS3 P32247 1/20 0.39
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
GRM4 Q14833 2/20 0.38
SYK P43405 1/20 0.38
PDCD1LG2 Q9BQ51 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30365211 1.00 CD274 (0.43) CD274PDCD1BRD4PTGER1XDH
SCHEMBL30364692 0.92 CD274 (0.51) CD274PDCD1BRD4RIPK1DHFR
SCHEMBL25149474 0.92 CD274 (0.51) CD274PDCD1BRD4RIPK1DHFR
SCHEMBL25149505 0.91 IRAK4 (0.46) CD274PDCD1BRD4DHFRDCPS
SCHEMBL25149242 0.90 PTGER1 (0.44) CD274PDCD1PTGER1RIPK1POLB
SCHEMBL30364967 0.90 PTGER1 (0.44) CD274PDCD1PTGER1RIPK1POLB
SCHEMBL30365021 0.82 CD274 (0.52) CD274PDCD1PTGER1RIPK1PDCD1LG2
SCHEMBL25149355 0.82 CD274 (0.52) CD274PDCD1PTGER1RIPK1PDCD1LG2
SCHEMBL30364797 0.82 CD274 (0.52) CD274PDCD1PTGER1RIPK1PDCD1LG2
SCHEMBL25149477 0.81 BRD4 (0.39) CD274PDCD1BRD4RIPK1GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023062575-A1 CYCLIC VINYL SULFONE COMPOUNDS AS WRN INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2023-04-20 WO disclosed