SCHEMBL25148786

SCHEMBL25148786

C/C(=C\C(C=O)=C(/NC=O)c1ccccc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
PARP15 Q460N3 1/20 0.42
PARP10 Q53GL7 1/20 0.42
CYP2C9 P11712 1/20 0.41
AKR1C3 P42330 1/20 0.39
ALDH1A1 P00352 5/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPT P10636 3/20 0.34
LMNA P02545 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25148649 0.90 ALDH1A1 (0.37) PARP1PARP15PARP10CYP2C9ALDH1A1
SCHEMBL25148634 0.82 PARP1 (0.42) PARP1PARP15PARP10CYP2C9AKR1C3
SCHEMBL25148694 0.78 PARP1 (0.39) PARP1PARP15PARP10CYP2C9AKR1C3
SCHEMBL13243496 0.77 ALDH1A1 (0.41) PARP1AKR1C3ALDH1A1MAPK1TDP1
SCHEMBL28533849 0.75 ALDH1A1 (0.40) PARP1ALDH1A1MAPK1TDP1MTNR1A
SCHEMBL5566136 0.70 AKR1C3 (0.54) PARP1PARP15PARP10CYP2C9AKR1C3
SCHEMBL2791186 0.69 NFE2L2 (0.59) PARP1PARP15PARP10CYP2C9AKR1C3
SCHEMBL8104632 0.69 NFE2L2 (0.59) PARP1PARP15PARP10CYP2C9AKR1C3
SCHEMBL25149538 0.69 ALDH1A1 (0.34) PARP1PARP15PARP10CYP2C9ALDH1A1
SCHEMBL3386465 0.68 AKR1C3 (0.50) PARP1PARP15PARP10CYP2C9AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023062575-A1 CYCLIC VINYL SULFONE COMPOUNDS AS WRN INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2023-04-20 WO disclosed