SCHEMBL25149261

SCHEMBL25149261

COc1nc(-c2ccccc2OCC2CCCCC2)ccc1C(=O)N[C@@H]1C=CS(=O)(=O)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
RIPK1 Q13546 4/20 0.39
IDH1 O75874 4/20 0.39
PTGER1 P34995 1/20 0.38
CD274 Q9NZQ7 2/20 0.37
PDCD1 Q15116 1/20 0.37
FAAH O00519 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
GUCY1B2 O75343 2/20 0.36
GUCY1A2 P33402 2/20 0.36
GUCY1A1 Q02108 2/20 0.36
GUCY1B1 Q02153 2/20 0.36
PDCD1LG2 Q9BQ51 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30365050 1.00 MEN1 (0.39) MEN1LMNAKMT2ARIPK1IDH1
SCHEMBL30364863 0.92 BRD4 (0.39) MEN1LMNAKMT2ARIPK1CD274
SCHEMBL25149477 0.92 BRD4 (0.39) MEN1LMNAKMT2ARIPK1CD274
SCHEMBL30364797 0.81 CD274 (0.52) RIPK1PTGER1CD274PDCD1FAAH
SCHEMBL30365021 0.81 CD274 (0.52) RIPK1PTGER1CD274PDCD1FAAH
SCHEMBL25149355 0.81 CD274 (0.52) RIPK1PTGER1CD274PDCD1FAAH
SCHEMBL25149242 0.80 PTGER1 (0.44) RIPK1PTGER1CD274PDCD1FAAH
SCHEMBL30364967 0.80 PTGER1 (0.44) RIPK1PTGER1CD274PDCD1FAAH
SCHEMBL30364997 0.78 LMNA (0.44) MEN1LMNAKMT2ACNR1CNR2
SCHEMBL30364609 0.73 LMNA (0.41) MEN1LMNAKMT2ACD274CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023062575-A1 CYCLIC VINYL SULFONE COMPOUNDS AS WRN INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2023-04-20 WO disclosed