SCHEMBL25164609

SCHEMBL25164609

Cc1cc(C(F)(F)F)nnc1C(C)C

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
CRHBP P24387 1/20 0.37
CYP2C19 P33261 1/20 0.37
CRHR2 Q13324 1/20 0.37
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16248172 0.78 CYP3A4 (0.36) CYP3A4CYP2D6TSHRCRHBPCYP2C19
SCHEMBL18307332 0.74 KDM4E (0.43) KDM4ELMNAHSP90AA1HSP90AB1
SCHEMBL31648936 0.72 KMT2A (0.43) KDM4ELMNACYP3A4CYP2D6TSHR
SCHEMBL30327770 0.71 KDM4E (0.41) KDM4ELMNAHSP90AA1HSP90AB1
SCHEMBL17688749 0.71 HSP90AA1 (0.44) KDM4ELMNAHSP90AA1HSP90AB1
SCHEMBL12848583 0.70 NOS3 (0.34)
SCHEMBL24542697 0.70 NOS2 (0.39)
SCHEMBL25928386 0.68
SCHEMBL24457882 0.68 KDM4E (0.39) KDM4ELMNACYP2C19HSP90AA1HSP90AB1
SCHEMBL24457884 0.68 KDM4E (0.39) KDM4ELMNACYP3A4CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064343-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2023-04-20 WO disclosed