Tolfenamic Acid

Tolfenamic Acid

SCHEMBL25190

Cc1c(Cl)cccc1Nc1ccccc1C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 8/20 1.00
PTGS2 P35354 5/20 1.00
MEN1 O00255 3/20 1.00
AKR1C3 P42330 3/20 1.00
KMT2A Q03164 3/20 1.00
LMNA P02545 2/20 1.00
CYP1A2 P05177 2/20 1.00
CYP3A4 P08684 2/20 1.00
CYP2C9 P11712 2/20 1.00
HIF1A Q16665 2/20 1.00
TTR P02766 2/20 1.00
ADORA3 P0DMS8 2/20 1.00
USP2 O75604 1/20 1.00
PLA2G1B P04054 1/20 1.00
PGR P06401 1/20 1.00
HTR1A P08908 1/20 1.00
ADRA2A P08913 1/20 1.00
AR P10275 1/20 1.00
MAPT P10636 1/20 1.00
HPGD P15428 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tolfenamic Acid SCHEMBL8060884 1.00 MT-CO2 (1.00) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL29389998 1.00 MT-CO2 (1.00) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL29484181 1.00 MT-CO2 (1.00) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL27540385 0.98 MT-CO2 (0.97) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL10619715 0.94 MT-CO2 (0.89) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL28095333 0.93 MT-CO2 (0.86) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL28229025 0.90 MT-CO2 (0.82) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL14976730 0.90 MT-CO2 (0.82) MT-CO2PTGS2MEN1AKR1C3KMT2A
SCHEMBL11564152 0.88 MT-CO2 (0.78) MT-CO2PTGS2MEN1AKR1C3KMT2A
SCHEMBL12608896 0.87 MT-CO2 (0.77) MT-CO2PTGS2MEN1AKR1C3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 21878 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
EP-4744663-A2 SKIN COMPOSITION Eaderm Co., Ltd. (JP) 2026-05-20 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-12605432-B2 Combinations for antigen based therapy DIAMYD MEDICAL AB (SE) 2026-04-21 US claimed
US-12600696-B2 Aromatic compounds Xeniopro GmbH (DE) 2026-04-14 US claimed
US-20260076961-A1 COMBINATION TREATMENTS Celex Oncology Innovations Limited (GB) 2026-03-19 US claimed
US-20260069532-A1 METHOD FOR MORSELIZING AND/OR TARGETING PHARMACEUTICALLY ACTIVE PRINCIPLES TO SYNOVIAL TISSUE MEDINCELL S.A. (FR) 2026-03-12 US claimed
US-12558309-B2 Method for morselizing and/or targeting pharmaceutically active principles to synovial tissue MEDINCELL S.A. (FR) 2026-02-24 US claimed
US-12545750-B2 Method for the diimide hydrogenation of emulsified unsaturated polymers PARKER DANE K (US) 2026-02-10 US claimed
EP-4680240-A1 METHOD OF TREATING DISORDERS WITH SURF1 MALFUNCTION Cure Mito Foundation (US) 2026-01-21 EP claimed
EP-0205492-A1 ANALGESIC, ANTI-INFLAMMATORY AND SKELETAL MUSCLE RELAXANT COMPOSITIONS SUNSHINE, Abraham (US) 1986-12-30 EP claimed
WO-1986003681-A1 ANALGESIC, ANTI-INFLAMMATORY AND SKELETAL MUSCLE RELAXANT COMPOSITIONS SUNSHINE ABRAHAM 1986-07-03 WO claimed
US-4594357-A Depot antiinflammatory agents TROPONWERKE GMBH & CO. (DE) 1986-06-10 US claimed
EP-0180597-A1 COUGH/COLD MIXTURES COMPRISING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS. SUNSHINE ABRAHAM (US) 1986-05-14 EP claimed
EP-0167566-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME SUNSHINE, Abraham (US) 1986-01-15 EP claimed
WO-1985004589-A1 COUGH/COLD MIXTURES COMPRISING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS SUNSHINE ABRAHAM 1985-10-24 WO claimed
WO-1985002542-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME SUNSHINE ABRAHAM 1985-06-20 WO claimed
EP-0130524-A2 Depot antiphlogistics Troponwerke GmbH & Co. KG (DE) 1985-01-09 EP claimed
EP-0114886-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE. SUNSHINE ABRAHAM (US) 1984-08-08 EP claimed
WO-1984000490-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE AND METHODS OF USING SAME SUNSHINE ABRAHAM 1984-02-16 WO claimed