Tolfenamic Acid

Tolfenamic Acid

SCHEMBL14976730

Cc1c(Cl)cccc1Nc1ccccc1C(=O)O.O=[As]O[As]=O

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 10/20 0.82
PTGS2 P35354 5/20 0.82
MEN1 O00255 3/20 0.82
AKR1C3 P42330 3/20 0.82
KMT2A Q03164 3/20 0.82
LMNA P02545 2/20 0.82
CYP1A2 P05177 2/20 0.82
CYP3A4 P08684 2/20 0.82
CYP2C9 P11712 2/20 0.82
HIF1A Q16665 2/20 0.82
TTR P02766 2/20 0.82
ADORA3 P0DMS8 2/20 0.82
USP2 O75604 1/20 0.82
PLA2G1B P04054 1/20 0.82
PGR P06401 1/20 0.82
HTR1A P08908 1/20 0.82
ADRA2A P08913 1/20 0.82
AR P10275 1/20 0.82
MAPT P10636 1/20 0.82
HPGD P15428 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tolfenamic Acid SCHEMBL8060884 0.90 MT-CO2 (1.00) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL25190 0.90 MT-CO2 (1.00) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL29389998 0.90 MT-CO2 (1.00) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL29484181 0.90 MT-CO2 (1.00) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL27540385 0.89 MT-CO2 (0.97) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL10619715 0.85 MT-CO2 (0.89) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL28095333 0.84 MT-CO2 (0.86) MT-CO2PTGS2MEN1AKR1C3KMT2A
Tolfenamic Acid SCHEMBL28229025 0.82 MT-CO2 (0.82) MT-CO2PTGS2MEN1AKR1C3KMT2A
SCHEMBL30593456 0.79 MT-CO2 (0.73) MT-CO2PTGS2MEN1AKR1C3KMT2A
SCHEMBL13465152 0.79 MT-CO2 (0.73) MT-CO2PTGS2MEN1AKR1C3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296716-B2 Androgen receptor ligands THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, & THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIV. TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2016-03-29 US disclosed
US-20140357682-A1 ANDROGEN RECEPTOR LIGANDS The Provost, Fellows, Foundation Scholars, & the Other Members of Board, of The College of the Holy (IE) 2014-12-04 US disclosed
EP-2782643-A1 ANDROGEN RECEPTOR LIGANDS The Provost, Fellows, Foundation Scholars, & the other members of Board, of the College of the Holy & Undiv. Trinity of Queen Elizabeth near Dublin (IE) 2014-10-01 EP disclosed
WO-2013076275-A1 ANDROGEN RECEPTOR LIGANDS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, & THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY & UNDIV.TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2013-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140357682-A1 ANDROGEN RECEPTOR LIGANDS AR, NR5A1, SHBG MT-CO2 3388/4885PTGS2 1012/4885MEN1 4657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.