SCHEMBL25192580

SCHEMBL25192580

CC(C)(C)[Si](C)(C)OCc1cnccc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 19/20 0.42
KDM6B O15054 6/20 0.41
KDM4E B2RXH2 3/20 0.41
KDM4A O75164 3/20 0.41
KDM4D Q6B0I6 3/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
BACE1 P56817 1/20 0.39
KDM5C P41229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31132807 1.00 KDM4C (0.42) KDM4CKDM6BKDM4EKDM4AKDM4D
Propionic Acid SCHEMBL29088348 0.85 TDP1 (0.39) KDM4CKDM6BKDM4EKDM4AKDM4D
Benzoic Acid SCHEMBL29088369 0.85 KDM4C (0.39) KDM4CKDM6BKDM4EKDM4AKDM4D
SCHEMBL31094071 0.81 BACE1 (0.49) MEN1ALDH1A1KMT2ABACE1
SCHEMBL6673753 0.81 BACE1 (0.49) MEN1ALDH1A1KMT2ABACE1
SCHEMBL1028187 0.79 KDM4C (0.49) KDM4CKDM6BKDM4EKDM4AKDM4D
SCHEMBL8528756 0.78 BACE1 (0.40) KDM4CKDM6BKDM4DMEN1ALDH1A1
SCHEMBL23199149 0.77 HDAC1 (0.40) TDP1BACE1
SCHEMBL15286291 0.76 BACE1 (0.38) KDM4CKDM4EALDH1A1MAPTTDP1
SCHEMBL14659892 0.76 AOC1 (0.37) KDM4EALDH1A1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4704830-A2 MRGPRX2 INHIBITORS AND METHODS OF USE THEREOF Septerna, Inc. (US) 2026-03-11 EP disclosed
WO-2024226914-A2 MRGPRX2 ANTAGONISTS AND METHODS OF USE THEREOF SEPTERNA, INC. (US) 2024-10-31 WO disclosed
CN-116472268-A Compounds capable of binding to proteins and conjugates obtained from these compounds MC SAF公司 2023-07-21 CN disclosed
EP-4181964-A1 COMPOUNDS CAPABLE OF BINDING TO PROTEINS AND CONJUGATES OBTAINED FROM THESE COMPOUNDS Mc SAF (FR) 2023-05-24 EP disclosed
CN-114173825-A Antibody-drug conjugates and their use in therapy MCSAF公司 2022-03-11 CN disclosed