SCHEMBL2520510

SCHEMBL2520510

CCOC(=O)c1cc2n(n1)CCNC2=O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.46
ADORA3 P0DMS8 1/20 0.40
RPS6KA3 P51812 1/20 0.40
ALDH1A1 P00352 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KMT2A Q03164 2/20 0.39
JMJD6 Q6NYC1 1/20 0.39
LMNA P02545 1/20 0.39
MMP2 P08253 1/20 0.39
MMP13 P45452 1/20 0.39
MMP14 P50281 1/20 0.39
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19902330 0.90 CDC7 (0.44) CDC7RPS6KA3ALDH1A1KMT2AJMJD6
SCHEMBL22716058 0.85 CDC7 (0.49) CDC7ADORA3ALDH1A1KMT2AJMJD6
SCHEMBL19902329 0.84 CDC7 (0.41) CDC7RPS6KA3ALDH1A1KMT2APIM1
SCHEMBL29256111 0.82 ALDH1A1 (0.70) ALDH1A1KMT2ALMNACYP1A2CYP2C19
SCHEMBL12092839 0.80 CDC7 (0.52) CDC7RPS6KA3ALDH1A1KMT2APIM1
SCHEMBL15009288 0.79 CDC7 (0.54) CDC7ALDH1A1PIM1PIM2SMN1; SMN2
SCHEMBL4192947 0.77 CDC7 (0.52) CDC7RPS6KA3ALDH1A1PIM1PIM2
SCHEMBL23980134 0.77 CYP1A2 (0.46) ADORA3ALDH1A1L3MBTL1KMT2ACYP1A2
SCHEMBL3127245 0.77 ALDH1A1 (0.46) CDC7ADORA3RPS6KA3ALDH1A1KMT2A
SCHEMBL6385372 0.77 CYP1A2 (0.44) ADORA3ALDH1A1L3MBTL1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 86 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12479831-B2 Substituted N(-methyl-D3)pyridazine-3-carboxamide or M-(methyl-D3)-nicotinamide compounds as IL-12, IL-23 and/or IFNα modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2025-11-25 US disclosed
US-20250270223-A1 CRYSTAL OF SUBSTITUTED PIPERAZINE DERIVATIVE AND PREPARATION METHOD THEREFOR Kangbaida (Sichuan) Biotechnology Co., Ltd (CN) 2025-08-28 US disclosed
EP-4504728-A1 PYRAZOLOPYRAZINONE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF Sanofi (FR) 2025-02-12 EP disclosed
US-20240383868-A1 SMARCA DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2024-11-21 US disclosed
CN-118946563-A Pyrazolopyrazinone compounds, process for their preparation and their therapeutic use 赛诺菲 2024-11-12 CN disclosed
CN-118434744-A Nitrogen-containing macrocyclic compound, and preparation method and medical application thereof 中国医药研究开发中心有限公司 2024-08-02 CN disclosed
US-20240158406-A1 PIPERAZINE DERIVATIVE AND USE THEREOF IN MEDICINE KANGBAIDA (SICHUAN) BIOTECHNOLOGY CO., LTD. (CN) 2024-05-16 US disclosed
EP-4342896-A1 PIPERAZINE DERIVATIVE AND USE THEREOF IN MEDICINE Chengdu Baiyu Pharmaceutical Co., Ltd. (CN) 2024-03-27 EP disclosed
CN-117586263-A Piperazine derivatives and their use in medicine 成都百裕制药股份有限公司 2024-02-23 CN disclosed
US-20240034723-A1 PIPERIDINYL SMALL MOLECULE DEGRADERS OF HELIOS AND METHODS OF USE DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-02-01 US disclosed
US-20120295913-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS VANDERBILT UNIVERSITY 2012-11-22 US disclosed
US-20120295913-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS VANDERBILT UNIVERSITY 2012-11-22 US disclosed
US-20120225844-A1 BICYCLIC TRIAZOLE AND PYRAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS JANSSEN-CILAG S.A. (ES) 2012-09-06 US disclosed
US-20120225844-A1 BICYCLIC TRIAZOLE AND PYRAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS JANSSEN-CILAG S.A. (ES) 2012-09-06 US disclosed
WO-2012083224-A1 BICYCLIC TRIAZOLE AND PYRAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS VANDERBILT UNIVERSITY (US) 2012-06-21 WO disclosed
WO-2012078817-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS VANDERBILT UNIVERSITY (US) 2012-06-14 WO disclosed
WO-2011130163-A1 SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-10-20 WO disclosed
WO-2011130163-A1 SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-10-20 WO disclosed
US-20110251184-A1 SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-10-13 US disclosed
US-20110251184-A1 SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250270223-A1 CRYSTAL OF SUBSTITUTED PIPERAZINE DERIVATIVE AND PREPARATION METHOD THEREFOR WEE1, WEE2, WASF2 CDC7 3034/4885ADORA3 4352/4885RPS6KA3 3714/4885
US-20110251184-A1 SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF HDAC6, HDAC1, H1-3 CDC7 3550/4885ADORA3 1818/4885RPS6KA3 1071/4885
US-12479831-B2 Substituted N(-methyl-D3)pyridazine-3-carboxamide or M-(methyl-D3)-nicotinamide compounds as IL-12, IL-23 and/or IFNα modulators TYK2, IRAK3, JAK3 CDC7 3419/4885ADORA3 324/4885RPS6KA3 246/4885
US-20240383868-A1 SMARCA DEGRADERS AND USES THEREOF SMARCA1, SMARCA2, SMARCC2 CDC7 1189/4885ADORA3 3738/4885RPS6KA3 2572/4885
US-20240034723-A1 PIPERIDINYL SMALL MOLECULE DEGRADERS OF HELIOS AND METHODS OF USE IKZF2, IKZF1, NUTF2 CDC7 3875/4885ADORA3 4616/4885RPS6KA3 4056/4885
US-20120225844-A1 BICYCLIC TRIAZOLE AND PYRAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS GRM5, GRIK5, GRIN3A CDC7 3768/4885ADORA3 139/4885RPS6KA3 908/4885
US-20240158406-A1 PIPERAZINE DERIVATIVE AND USE THEREOF IN MEDICINE VHL, GLS2, GOT2 CDC7 4657/4885ADORA3 2786/4885RPS6KA3 1435/4885
US-20120295913-A1 BICYCLIC PYRAZOLE COMPOUNDS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS GRM5, GRIK5, GRM3 CDC7 4213/4885ADORA3 120/4885RPS6KA3 1630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.