Formamide

Formamide

SCHEMBL252132

Cc1ccc(Br)cc1-n1cnc(C(N)=O)c1-c1nc2cccc(OC3CCN(C)CC3)c2[nH]1.NC=O

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.37
NEK2 P51955 9/20 0.34
PLK1 P53350 7/20 0.34
BRD4 O60885 1/20 0.34
PDGFRB P09619 2/20 0.32
KDR P35968 2/20 0.32
FGFR1 P11362 1/20 0.32
PIK3CD O00329 1/20 0.31
NUAK1 O60285 1/20 0.31
PIM1 P11309 1/20 0.31
PLK3 Q9H4B4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL216161 0.84 NEK2 (0.33) CHEK2NEK2PLK1KDR
SCHEMBL215858 0.76 TOP2A (0.35)
SCHEMBL213660 0.74 TOP2A (0.35)
SCHEMBL216162 0.69 ALDH1A1 (0.39) KDRL3MBTL1
SCHEMBL214572 0.65 BTK (0.42) KDR
SCHEMBL214751 0.65 BTK (0.38) KDR
SCHEMBL27040144 0.64 AMY1A (0.47) CHEK2BRD4PDGFRBKDRFGFR1
SCHEMBL214823 0.62 CHEK2 (0.35) CHEK2PLK1PLK3
SCHEMBL214920 0.62 MAPK14 (0.42)
Hydrochloric Acid SCHEMBL213800 0.62 CHEK2 (0.35) CHEK2PLK1PLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088767-B2 JAK-2 modulators and methods of use EXELIXIS, INC. (US) 2012-01-03 US claimed