SCHEMBL25216352

SCHEMBL25216352

CCCn1cc(C(=O)O)nc1CC

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
CYP19A1 P11511 1/20 0.38
BRD4 O60885 1/20 0.36
HCAR2 Q8TDS4 2/20 0.35
TYR P14679 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
PTGER1 P34995 1/20 0.33
KDM5A P29375 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
CNR2 P34972 2/20 0.32
CYP2C19 P33261 1/20 0.32
PLA2G4A P47712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28218206 0.88 CYP19A1 (0.37) L3MBTL1CYP19A1BRD4HCAR2RXFP1
SCHEMBL16519369 0.80 PTGER1 (0.42) L3MBTL1CYP19A1BRD4HCAR2RXFP1
SCHEMBL28896966 0.79 CYP19A1 (0.32) CYP19A1BRD4
SCHEMBL28314805 0.79 L3MBTL1 (0.40) L3MBTL1BRD4HCAR2TYRRXFP1
SCHEMBL4934202 0.78 HCAR2 (0.43) L3MBTL1HCAR2CYP2C19PLA2G4A
SCHEMBL29094923 0.75 HCAR2 (0.37) L3MBTL1CYP19A1HCAR2RXFP1PTGS1
SCHEMBL21564316 0.74 HCAR2 (0.41) L3MBTL1BRD4HCAR2RXFP1PTGS1
SCHEMBL15903278 0.72 HCAR2 (0.35) CYP19A1HCAR2RXFP1PTGS1PTGS2
SCHEMBL6494245 0.72 RXFP1 (0.36) L3MBTL1BRD4HCAR2RXFP1PTGS1
SCHEMBL1268994 0.70 WDR5 (0.36) CYP19A1HCAR2RXFP1PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12583849-B2 KCNT1 inhibitors and methods of use PRAXIS PRECISION MEDICINES, INC. (US) 2026-03-24 US disclosed
EP-4692069-A2 KCNT1 INHIBITORS AND METHODS OF USE Praxis Precision Medicines, Inc. (US) 2026-02-11 EP disclosed
EP-4110317-B1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PREC MEDICINES INC (US) 2025-11-19 EP disclosed
US-20230167102-A1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PRECISION MEDICINES, INC. 2023-06-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12583849-B2 KCNT1 inhibitors and methods of use KCNT1, SCN1A, KCNT2 L3MBTL1 296/4885CYP19A1 3935/4885BRD4 2646/4885
US-20230167102-A1 KCNT1 INHIBITORS AND METHODS OF USE KCNT1, KCNT2, KCNQ2 L3MBTL1 656/4885CYP19A1 3818/4885BRD4 1366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.