SCHEMBL2522333

SCHEMBL2522333

COc1ccc(-c2ccc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)cn1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 14/20 0.80
LRRK2 Q5S007 3/20 0.58
CYP3A4 P08684 3/20 0.55
CYP2D6 P10635 2/20 0.55
CYP2C9 P11712 1/20 0.55
TDO2 P48775 1/20 0.54
DYRK1A Q13627 4/20 0.53
DYRK2 Q92630 3/20 0.53
DYRK1B Q9Y463 3/20 0.53
CLK1 P49759 1/20 0.53
DYRK3 O43781 1/20 0.49
CCNT1 O60563 1/20 0.49
CDK9 P50750 1/20 0.49
CDK5 Q00535 1/20 0.49
CDK5R1 Q15078 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.47
SGK1 O00141 1/20 0.46
IKBKB O14920 1/20 0.46
AURKA O14965 1/20 0.46
CHUK O15111 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL721794 0.89 MAP3K11 (1.00) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL7328650 0.88 MAP3K11 (0.70) MAP3K11LRRK2TDO2DYRK1ADYRK2
SCHEMBL2527600 0.81 MAP3K11 (0.73) MAP3K11LRRK2DYRK1AKIT
SCHEMBL15759024 0.80 MAP3K11 (0.60) MAP3K11LRRK2CYP3A4CYP2D6TDO2
SCHEMBL2526092 0.78 MAP3K11 (0.60) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL7089345 0.77 MAP3K11 (0.56) MAP3K11TDO2DYRK1ADYRK2DYRK1B
SCHEMBL720862 0.76 MAP3K11 (1.00) MAP3K11LRRK2CYP3A4CYP2D6DYRK1A
SCHEMBL723789 0.76 MAP3K11 (1.00) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL2526465 0.76 NPC1 (0.71) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL724259 0.74 MAP3K11 (0.83) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379561-A2 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2011-10-26 EP disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed