SCHEMBL2526465

SCHEMBL2526465

c1ccc(-c2ccc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.71
MAP3K11 Q16584 7/20 0.68
DYRK1A Q13627 2/20 0.53
DYRK2 Q92630 2/20 0.53
DYRK1B Q9Y463 2/20 0.53
CYP3A4 P08684 2/20 0.50
CYP2D6 P10635 2/20 0.50
PIM1 P11309 2/20 0.50
PIM3 Q86V86 2/20 0.50
CLK1 P49759 1/20 0.50
CYP2C9 P11712 1/20 0.49
LRRK2 Q5S007 1/20 0.49
CASP3 P42574 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
GLO1 Q04760 1/20 0.47
IMPDH2 P12268 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL940968 0.86 MAP3K11 (0.58) NPC1MAP3K11DYRK1ADYRK2DYRK1B
SCHEMBL18552198 0.84 IMPDH2 (0.61) NPC1MAP3K11DYRK1APIM1PIM3
SCHEMBL18552149 0.84 IMPDH2 (0.61) NPC1MAP3K11DYRK1APIM1PIM3
SCHEMBL24022684 0.84 IMPDH2 (0.61) NPC1MAP3K11DYRK1APIM1PIM3
SCHEMBL446619 0.84 NPC1 (1.00) NPC1MAP3K11DYRK1ADYRK2DYRK1B
SCHEMBL30587350 0.84 NPC1 (1.00) NPC1MAP3K11DYRK1ADYRK2DYRK1B
SCHEMBL28210414 0.82 NPC1 (0.96) NPC1MAP3K11DYRK1ADYRK2DYRK1B
SCHEMBL721629 0.81 MAP3K11 (1.00) MAP3K11DYRK1ADYRK2DYRK1BCYP3A4
SCHEMBL20120884 0.81 NPC1 (0.92) NPC1MAP3K11DYRK1ADYRK2DYRK1B
SCHEMBL2527600 0.80 MAP3K11 (0.73) NPC1MAP3K11DYRK1ALRRK2CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379561-A2 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2011-10-26 EP disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed