SCHEMBL2523004

SCHEMBL2523004

C=CC(=O)OCCN(CCCC)S(=O)(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.46
HPGD P15428 1/20 0.46
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 1/20 0.36
THRB P10828 1/20 0.35
TP53 P04637 2/20 0.33
HIF1A Q16665 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MMP1 P03956 2/20 0.32
MMP2 P08253 2/20 0.32
MMP9 P14780 2/20 0.32
MMP8 P22894 2/20 0.32
MMP13 P45452 2/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
ATM Q13315 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31127917 1.00 TSHR (0.46) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL633255 0.94 TSHR (0.40) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL30424942 0.93 TSHR (0.38) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL560589 0.90 TSHR (0.38) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL7920244 0.90 TSHR (0.38) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL9873897 0.90 TSHR (0.38) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL7920243 0.90 TSHR (0.38) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL7906773 0.89 TSHR (0.39) TSHRHPGDALDH1A1CYP3A4THRB
SCHEMBL4669429 0.83 TSHR (0.43) TSHRTHRBMMP1MMP2MMP9
SCHEMBL16178607 0.83 TSHR (0.36) TSHRHPGDALDH1A1CYP3A4THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 291 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039093-B2 Method for preparing tamperproof ID documents AGFA-GEVAERT N.V. (BE) 2011-10-18 US claimed
WO-2009080626-A2 TAMPERPROOF SECURITY DOCUMENT AND PROCESS FOR PREPARING TAMPERPROOF SECURITY DOCUMENTS AGFA-GEVAERT NV (BE) 2009-07-02 WO claimed
EP-0914079-B2 HAIR SHAMPOO COMPRISING SILICONE COMPOUNDS OREAL (FR) 2009-07-01 EP claimed
WO-2009077536-A2 PROCESS FOR PREPARING TAMPERPROOF SECURITY DOCUMENTS AND TAMPERPROOF SECURITY DOCUMENT AGFA-GEVAERT NV (BE) 2009-06-25 WO claimed
EP-1940981-A1 METHOD FOR PREPARING TAMPERPROOF ID DOCUMENTS AGFA-GEVAERT N.V. (BE) 2008-07-09 EP claimed
US-20070092703-A1 Method for preparing tamperproof ID documents AGFA-GEVAERT (BE) 2007-04-26 US claimed
WO-2007045578-A1 METHOD FOR PREPARING TAMPERPROOF ID DOCUMENTS AGFA-GEVAERT (BE) 2007-04-26 WO claimed
EP-1029030-B1 FOAMING-RESISTANT HYDROCARBON OIL COMPOSITIONS SOLUTIA INC (US) 2003-01-15 EP claimed
US-6503494-B1 Cosmetic or dermatological composition for treating hair; improved feel such as softness and smoothness L'OREAL S.A. (FR) 2003-01-07 US claimed
EP-0853470-B1 COSMETIC COMPOSITION INCLUDING AT LEAST ONE SILICONE-GRAFTED POLYMER AND AT LEAST ONE COMBINATION OF AN ANIONIC POLYMER AND A CATIONIC POLYMER OREAL (FR) 2002-12-04 EP claimed
US-6090376-A CONSISTS OF A GRAFTED SILICON POLYMER WITH A NON-SILICON POLYMER GRAFTED BY ONE POLYSILOXANE MONOMER AND ATLEAST ONE IONIC AMPHIPHILIC POLYMER CONSISTING OF A FATTY CHAIN AND ATLEAST ONE HYDROPHILIC UNIT; COSMETIC L'OREAL (FR) 2000-07-18 US claimed
US-6011126-A HAIR CONDITIONERS L'OREAL (FR) 2000-01-04 US claimed
WO-1999020721-A1 FOAMING-RESISTANT HYDROCARBON OIL COMPOSITIONS SOLUTIA INC. (US) 1999-04-29 WO claimed
EP-0773016-B1 Topical composition containing a combination of a silicon grafted polymer with a non-silicon backbone and a non-silicon grafted polysiloxan polymer OREAL (FR) 1998-04-01 EP claimed
EP-0333464-B1 POLYMER CLADDINGS FOR OPTICAL FIBRE WAVEGUIDES MINNESOTA MINING & MFG (US) 1993-05-12 EP claimed
US-5152287-A Cross-linked fluorinated polymers for use in gas sensors CORDIS CORPORATION (US) 1992-10-06 US claimed
US-4968116-A HEAT RESISTANCE MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1990-11-06 US claimed
US-4957982-A PROTECTIVE COATED SURFACES CROWN DECORATIVE PRODUCTS LIMITED (GB) 1990-09-18 US claimed
EP-0333464-A1 Polymer claddings for optical fibre waveguides MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1989-09-20 EP claimed
EP-0307074-A2 Antifouling coating for polymerisation reactors Crown Berger Limited (GB) 1989-03-15 EP claimed