SCHEMBL25239407

SCHEMBL25239407

O=C(O)c1cncc(-c2cc(Cl)ccc2Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.56
MKNK1 Q9BUB5 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
TBXA2R P21731 1/20 0.49
PTGER1 P34995 1/20 0.49
ALDH1A1 P00352 2/20 0.49
TP53 P04637 1/20 0.49
SRD5A2 P31213 1/20 0.45
POLB P06746 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 1/20 0.43
DDO Q99489 1/20 0.43
SCN2A Q99250 1/20 0.43
SCN10A Q9Y5Y9 1/20 0.43
MAP4K4 O95819 1/20 0.43
CTSA P10619 1/20 0.42
CNR2 P34972 1/20 0.42
P2RX7 Q99572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28238707 0.84 CTSA (0.53) HCAR2MKNK1MKNK2TBXA2RPTGER1
SCHEMBL1840398 0.81 MKNK1 (0.68) HCAR2MKNK1MKNK2SCN2ASCN10A
SCHEMBL3072205 0.81 ALPL (0.57) HCAR2MKNK1MKNK2TBXA2RPTGER1
SCHEMBL2050887 0.80 SRD5A2 (0.68) PTGER1ALDH1A1TP53SRD5A2KDM4E
SCHEMBL29788156 0.80 SRD5A2 (0.68) PTGER1ALDH1A1TP53SRD5A2KDM4E
SCHEMBL30775592 0.79 MKNK1 (0.59) HCAR2MKNK1MKNK2SRD5A2KDM4E
SCHEMBL25234831 0.79 CYP2C9 (0.54) ALDH1A1POLBKDM4ELMNACTSA
SCHEMBL4401794 0.77 RXRA (0.58) HCAR2MKNK1MKNK2MAP4K4
SCHEMBL3181717 0.76 MKNK1 (0.69) HCAR2MKNK1MKNK2ALDH1A1POLB
SCHEMBL14691606 0.76 KMO (0.49) HCAR2MKNK1MKNK2CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023114977-A1 S1PR4 RECEPTOR ANTAGONISTS AND METHODS OF USE THEREOF TIAKI THERAPEUTICS, INC. (US) 2023-06-22 WO disclosed