SCHEMBL2524802

SCHEMBL2524802

CCC(C(=O)O)C1C(=O)Nc2cc(O)ccc21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.34
TDO2 P48775 2/20 0.34
MAOB P27338 1/20 0.32
CYP2C9 P11712 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ESR1 P03372 2/20 0.31
ESR2 Q92731 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
SLC10A2 Q12908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1899980 0.73 PGR (0.40) IDO1TDO2MAOBKMT2AMEN1
SCHEMBL562407 0.71 CYP1A2 (0.56) CYP2C9HSD17B10ESR1ESR2KMT2A
SCHEMBL2878152 0.70 EGFR (0.44) IDO1TDO2HSD17B10ALDH1A1MAPT
SCHEMBL27986400 0.70 PGR (0.45) MAOBCYP2C9HSD17B10ESR1ESR2
SCHEMBL10562450 0.66 MAOB (0.50) IDO1MAOBESR1ESR2MAPT
SCHEMBL2887312 0.66 CDYL2 (0.42) IDO1TDO2HSD17B10MAPTKMT2A
SCHEMBL1400719 0.66 ESR1 (0.61) ESR1ESR2
SCHEMBL820847 0.66 ESR1 (0.61) ESR1ESR2
SCHEMBL5789865 0.66 ESR1 (0.61) ESR1ESR2
SCHEMBL820547 0.66 ESR1 (0.61) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039484-B2 Antidiabetic bicyclic compounds MERCK SHARP & DOHME CORP. (US) 2011-10-18 US disclosed