SCHEMBL25254475

SCHEMBL25254475

CCCCC(=O)Nc1cnc2ccsc2c1NCC1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 18/20 0.55
CYP2D6 P10635 4/20 0.49
CYP2C9 P11712 4/20 0.49
CYP3A4 P08684 3/20 0.49
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31025948 1.00 GRIN2B (0.55) GRIN2BCYP2D6CYP2C9CYP3A4MEN1
SCHEMBL29030555 0.87 NPC1 (0.37) GRIN2BCYP2C9MEN1LMNAKMT2A
SCHEMBL25299136 0.86 GPR119 (0.43)
SCHEMBL31025943 0.83 GRIN2B (0.65) GRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL25256028 0.83 GRIN2B (0.65) GRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL25301684 0.80 NPC1 (0.38) CYP2C9
SCHEMBL31270671 0.80 GRIN2B (0.60) GRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL25253285 0.80 GRIN2B (0.60) GRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL25294483 0.79 GRIN2B (0.38) GRIN2BCYP2D6CYP2C9CYP3A4MEN1
SCHEMBL25301779 0.77 KDM4E (0.42) GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023207710-A1 ANTIBODY-DRUG CONJUGATE, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2023-11-02 WO disclosed
WO-2023125121-A1 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2023-07-06 WO disclosed