SCHEMBL25294483

SCHEMBL25294483

COCCC(=O)Nc1cnc2ccsc2c1NCC1CCN(C(=O)O)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 7/20 0.38
BRD4 O60885 1/20 0.35
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
DRD3 P35462 1/20 0.34
ADORA2B P29275 3/20 0.34
ADORA2A P29274 2/20 0.34
NPY5R Q15761 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CASP3 P42574 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
MELK Q14680 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31270804 0.89 KDM4E (0.42) GRIN2BBRD4ADORA2BADORA2A
SCHEMBL25301779 0.89 KDM4E (0.42) GRIN2BBRD4ADORA2BADORA2A
SCHEMBL29030555 0.89 NPC1 (0.37) GRIN2BADORA2ANPY5RMEN1KMT2A
SCHEMBL25299136 0.79 GPR119 (0.43) ADORA2BADORA2A
SCHEMBL25254475 0.79 GRIN2B (0.55) GRIN2BMEN1KMT2ACYP3A4CYP2D6
SCHEMBL31025948 0.79 GRIN2B (0.55) GRIN2BMEN1KMT2ACYP3A4CYP2D6
SCHEMBL29030594 0.79 GRIN2B (0.44) GRIN2BADORA2BADORA2ACYP3A4CYP2D6
SCHEMBL25257180 0.77 MAPK8 (0.36) ADORA2BADORA2AMEN1KMT2A
SCHEMBL29030581 0.75 GRIN2B (0.39) GRIN2BADORA2BCYP3A4CYP2D6CYP2C9
SCHEMBL25301684 0.75 NPC1 (0.38) ADORA2BADORA2AL3MBTL1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125121-A1 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2023-07-06 WO disclosed