SCHEMBL2525751

SCHEMBL2525751

Cc1ccccc1OC[C@H]1CO1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 1.00
GLA P06280 1/20 1.00
TDP1 Q9NUW8 2/20 0.58
PKM P14618 2/20 0.58
TP53 P04637 3/20 0.52
TSHR P16473 3/20 0.52
HIF1A Q16665 2/20 0.52
CYP3A4 P08684 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
MAPT P10636 3/20 0.46
HPGD P15428 2/20 0.46
CYP1A2 P05177 2/20 0.46
PPARG P37231 1/20 0.46
ADRB2 P07550 1/20 0.45
HTR1A P08908 1/20 0.45
SLC6A2 P23975 1/20 0.45
HTR2A P28223 1/20 0.45
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2527037 1.00 ALDH1A1 (1.00) ALDH1A1GLATDP1PKMTP53
SCHEMBL29498775 1.00 ALDH1A1 (1.00) ALDH1A1GLATDP1PKMTP53
SCHEMBL179950 1.00 ALDH1A1 (1.00) ALDH1A1GLATDP1PKMTP53
SCHEMBL29424137 1.00 ALDH1A1 (1.00) ALDH1A1GLATDP1PKMTP53
Water SCHEMBL28245542 0.98 ALDH1A1 (0.96) ALDH1A1GLATDP1PKMTP53
Methane SCHEMBL28274836 0.98 ALDH1A1 (0.96) ALDH1A1GLATDP1PKMTP53
Propane SCHEMBL28104053 0.96 ALDH1A1 (0.93) ALDH1A1GLATDP1PKMTP53
SCHEMBL22653916 0.95 ALDH1A1 (0.90) ALDH1A1GLATDP1PKMTP53
Propylene Oxide SCHEMBL28819413 0.95 ALDH1A1 (0.90) ALDH1A1GLATDP1PKMTP53
SCHEMBL425554 0.92 ALDH1A1 (0.84) ALDH1A1GLATDP1PKMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114854714-A Kidney bean source epoxide hydrolase mutant, gene, vector, engineering bacterium, preparation method and application 安徽工程大学 2022-08-05 CN disclosed
CN-107189970-B Pseudomonas adynaudiana YC1612 for producing halohydrin dehalogenase and application and preparation method thereof 盐城工学院 2020-03-06 CN disclosed
CN-107189970-A A kind of cloudy city pseudomonad YC1612 and its application and preparation method for producing halide alcohol dehalogenase 盐城工学院 2017-09-22 CN disclosed
US-8039503-B2 Lapachone compounds and methods of use thereof ARQULE, INC. (US) 2011-10-18 US disclosed
US-20110105470-A1 Novel Lapachone Compounds And Methods of Use Thereof ARQULE, INC. (US) 2011-05-05 US disclosed
US-7902354-B2 Lapachone compounds and methods of use thereof ARQULE, INC. (US) 2011-03-08 US disclosed
US-20090105166-A1 Novel lapachone compounds and methods of use thereof ARQULE, INC. 2009-04-23 US disclosed
EP-2035435-A1 NOVEL LAPACHONE COMPOUNDS AND METHODS OF USE THEREOF ARQULE, INC. (US) 2009-03-18 EP disclosed
WO-2007139569-A1 NOVEL LAPACHONE COMPOUNDS AND METHODS OF USE THEREOF ARQULE, INC. (US) 2007-12-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105470-A1 Novel Lapachone Compounds And Methods of Use Thereof BAD, NQO1, CASP3 ALDH1A1 906/4885GLA 606/4885TDP1 2203/4885
US-20090105166-A1 Novel lapachone compounds and methods of use thereof BAD, NQO1, CASP3 ALDH1A1 906/4885GLA 606/4885TDP1 2203/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.