SCHEMBL25257948

SCHEMBL25257948

CC(C)NC(=O)Cc1cccc(Br)c1

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.58
EGFR P00533 5/20 0.54
ERBB2 P04626 5/20 0.54
MAPK8 P45983 1/20 0.49
GLS O94925 1/20 0.49
HSD17B10 Q99714 1/20 0.48
CNR2 P34972 1/20 0.48
SIGMAR1 Q99720 1/20 0.47
LMNA P02545 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27477588 0.85 EGFR (0.49) PTGESEGFRERBB2MAPK8GLS
SCHEMBL15065815 0.82 NLRP3 (0.50) CNR2SIGMAR1
SCHEMBL6136809 0.82 EGFR (0.52) PTGESEGFRERBB2MAPK8GLS
SCHEMBL5690915 0.81 EGFR (0.57) EGFRERBB2MAPK8GLSSIGMAR1
SCHEMBL1632800 0.81 GLS (0.49) GLSCNR2KMT2A
SCHEMBL12880514 0.81 EPHX2 (0.58) MAPK8CNR2SIGMAR1KMT2A
SCHEMBL11626990 0.80 EGFR (0.50) PTGESEGFRERBB2MAPK8GLS
SCHEMBL4057391 0.80 POLB (0.52) PTGESEGFRERBB2HSD17B10CNR2
SCHEMBL5871721 0.80 KMT2A (0.69) EGFRERBB2CNR2LMNAKMT2A
SCHEMBL15831226 0.79 POLB (0.58) PTGESMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250136552-A1 ANTAGONISTS OF CAV 2.3 LARIO THERAPEUTICS LIMITED (GB) 2025-05-01 US disclosed
EP-4436664-A1 ANTAGONISTS OF CAV 2.3 Lario Therapeutics Limited (GB) 2024-10-02 EP disclosed
WO-2023094828-A1 ANTAGONISTS OF CAV 2.3 LARIO THERAPEUTICS LIMITED (GB) 2023-06-01 WO disclosed
WO-2023094828-A1 ANTAGONISTS OF CAV 2.3 LARIO THERAPEUTICS LIMITED (GB) 2023-06-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250136552-A1 ANTAGONISTS OF CAV 2.3 CACNA1E, CACNA1A, CACNA1S PTGES 3444/4885EGFR 3545/4885ERBB2 1356/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.