SCHEMBL25258087

SCHEMBL25258087

COc1cc(C#N)cc2nc(N)n(CCc3ccc(Br)cc3)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
GAA P10253 4/20 0.41
KMT2A Q03164 4/20 0.41
MAPT P10636 4/20 0.41
KDM4E B2RXH2 3/20 0.41
HPGD P15428 2/20 0.41
ALOX15 P16050 2/20 0.41
CASP1 P29466 2/20 0.41
CASP7 P55210 2/20 0.41
HSD17B10 Q99714 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.37
GLA P06280 3/20 0.36
MEN1 O00255 1/20 0.36
CSF1R P07333 6/20 0.35
THRB P10828 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
NOD2 Q9HC29 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30581458 1.00 ALDH1A1 (0.41) ALDH1A1GAAKMT2AMAPTKDM4E
SCHEMBL25255010 0.89 ALDH1A1 (0.41) ALDH1A1GAAKMT2AMAPTKDM4E
SCHEMBL30581404 0.89 ALDH1A1 (0.41) ALDH1A1GAAKMT2AMAPTKDM4E
SCHEMBL30586471 0.86 CA2 (0.44) ALDH1A1GAAKMT2AMAPTKDM4E
SCHEMBL25251145 0.86 CA2 (0.44) ALDH1A1GAAKMT2AMAPTKDM4E
SCHEMBL25259879 0.80 STING1 (0.47) MAPT
SCHEMBL30581457 0.80 STING1 (0.47) MAPT
SCHEMBL25302212 0.78 KMT2A (0.47) ALDH1A1GAAKMT2AKDM4EGLA
SCHEMBL25262670 0.77 SMN1; SMN2 (0.44) ALDH1A1GAAKMT2AMAPTKDM4E
SCHEMBL30586457 0.77 SMN1; SMN2 (0.44) ALDH1A1GAAKMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116444544-A Benzimidazole compound and medical application thereof 中国科学院上海药物研究所 2023-07-18 CN disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed