SCHEMBL25259768

SCHEMBL25259768

COc1cc(C(N)=O)cc2nc(N)n(Cc3ccc(S(N)(=O)=O)cc3)c12

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.47
ENPP1 P22413 2/20 0.46
TSHR P16473 1/20 0.44
CA2 P00918 9/20 0.42
CA1 P00915 8/20 0.42
CA9 Q16790 6/20 0.42
CA14 Q9ULX7 2/20 0.42
USP2 O75604 1/20 0.42
CA7 P43166 1/20 0.42
CA12 O43570 2/20 0.41
STING1 Q86WV6 4/20 0.40
CA4 P22748 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30586480 1.00 KIF11 (0.47) KIF11ENPP1TSHRCA2CA1
SCHEMBL30586485 0.90 TSHR (0.48) KIF11TSHRCA2CA1CA9
SCHEMBL25258702 0.90 TSHR (0.48) KIF11TSHRCA2CA1CA9
SCHEMBL30586478 0.88 CA2 (0.44) ENPP1TSHRCA2CA1CA9
SCHEMBL25257071 0.88 CA2 (0.44) ENPP1TSHRCA2CA1CA9
SCHEMBL25259734 0.82 CA2 (0.39) ENPP1CA2CA1CA9CA7
SCHEMBL30586469 0.82 CA2 (0.39) ENPP1CA2CA1CA9CA7
SCHEMBL25253344 0.79 CA2 (0.43) TSHRCA2CA1CA9USP2
SCHEMBL30586476 0.79 CA2 (0.43) TSHRCA2CA1CA9USP2
SCHEMBL19437658 0.79 STING1 (0.52) ENPP1STING1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116444544-A Benzimidazole compound and medical application thereof 中国科学院上海药物研究所 2023-07-18 CN disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed