SCHEMBL25258702

SCHEMBL25258702

COc1cc(C(N)=O)cc2nc(N)n(CCc3ccc(S(N)(=O)=O)cc3)c12

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
KIF11 P52732 2/20 0.45
USP2 O75604 1/20 0.45
CA2 P00918 12/20 0.45
CA1 P00915 10/20 0.43
CA12 O43570 6/20 0.43
CA9 Q16790 6/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
MAPT P10636 1/20 0.43
CA4 P22748 2/20 0.41
STING1 Q86WV6 2/20 0.41
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30586485 1.00 TSHR (0.48) TSHRKIF11USP2CA2CA1
SCHEMBL25259768 0.90 KIF11 (0.47) TSHRKIF11USP2CA2CA1
SCHEMBL30586480 0.90 KIF11 (0.47) TSHRKIF11USP2CA2CA1
SCHEMBL25253344 0.89 CA2 (0.43) TSHRUSP2CA2CA1CA12
SCHEMBL30586476 0.89 CA2 (0.43) TSHRUSP2CA2CA1CA12
SCHEMBL25259879 0.87 STING1 (0.47) MAPTSTING1
SCHEMBL30581457 0.87 STING1 (0.47) MAPTSTING1
SCHEMBL30586471 0.82 CA2 (0.44) CA2CA1CA12CA9MAPT
SCHEMBL25251145 0.82 CA2 (0.44) CA2CA1CA12CA9MAPT
SCHEMBL19437552 0.80 STING1 (0.52) USP2STING1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116444544-A Benzimidazole compound and medical application thereof 中国科学院上海药物研究所 2023-07-18 CN disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed