SCHEMBL25263246

SCHEMBL25263246

COc1ncccc1-c1cc(C)ncc1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.50
POLQ O75417 14/20 0.48
EIF4E P06730 1/20 0.45
BTK Q06187 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
GPBAR1 Q8TDU6 1/20 0.40
ELANE P08246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25309592 0.88 POLQ (0.50) DHODHPOLQ
SCHEMBL7899073 0.83 DHODH (0.56) DHODHEIF4EBTK
SCHEMBL22717424 0.81 POLQ (0.60) DHODHPOLQ
SCHEMBL29574532 0.81 POLQ (0.60) DHODHPOLQ
SCHEMBL29575107 0.81 POLQ (0.60) DHODHPOLQ
SCHEMBL24501328 0.80 KDM4E (0.44) DHODHPOLQ
SCHEMBL29695223 0.80 KDM4E (0.44) DHODHPOLQ
SCHEMBL24770211 0.79 POLQ (0.60) POLQ
SCHEMBL30016080 0.79 POLQ (0.60) POLQ
SCHEMBL30905040 0.78 POLQ (0.45) POLQFFAR4GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250122221-A1 SIX-MEMBERED CYCLOTHIAZOLE COMPOUND AND USE THEREOF NANJING ZAIMING PHARMACEUTICAL CO., LTD. (CN) 2025-04-17 US disclosed
EP-4464709-A1 SIX-MEMBERED CYCLOTHIAZOLE COMPOUND AND USE THEREOF Nanjing Zaiming Pharmaceutical Co., Ltd. (CN) 2024-11-20 EP disclosed
CN-118525025-A Six-membered cyclothiazole compound and application thereof 南京再明医药有限公司 2024-08-20 CN disclosed
WO-2023134739-A1 SIX-MEMBERED CYCLOTHIAZOLE COMPOUND AND USE THEREOF 南京再明医药有限公司 2023-07-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250122221-A1 SIX-MEMBERED CYCLOTHIAZOLE COMPOUND AND USE THEREOF POLRMT, POLQ, POLH DHODH 236/4885POLQ 2/4885EIF4E 1203/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.