SCHEMBL25280494

SCHEMBL25280494

COC(=O)c1cnc2[nH]ccc2c1I

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AXL P30530 6/20 0.46
NUDT1 P36639 1/20 0.46
MAP2K1 Q02750 1/20 0.46
TTBK1 Q5TCY1 1/20 0.45
TTBK2 Q6IQ55 1/20 0.45
JAK3 P52333 9/20 0.43
JAK1 P23458 8/20 0.43
CDK8 P49336 1/20 0.42
PRKCI P41743 1/20 0.41
JAK2 O60674 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2632955 0.83 NUDT1 (0.50) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL31403755 0.83 NUDT1 (0.50) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL30985188 0.82 AXL (0.55) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL21632535 0.82 JAK3 (0.46) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL31403683 0.82 JAK3 (0.46) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL28798529 0.82 TTBK1 (0.48) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL29656385 0.82 TTBK1 (0.48) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL2115690 0.82 AXL (0.55) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL16940954 0.81 JAK3 (0.50) AXLNUDT1MAP2K1TTBK1TTBK2
SCHEMBL24455454 0.79 JAK3 (0.51) AXLNUDT1MAP2K1TTBK1TTBK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed